Isidakamizwa i-Alpha-lipon: imiyalo esetshenzisiwe

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I-Alphon Lipon isidakamizwa esinikeza ukuguquguquka kwezinqubo ze-metabolic. Ngaphansi kwethonya lesakhi esisebenzayo, kusetshenziswa ukusebenza okuzinzile kwezitho zepheshana lesisu. Isetshenziselwa ukwelapha isifo sikashukela i-neuropathy.

Igama Lezwe elingafanele

Ukulungiselela kwe-INN: i-alpha lipoic acid.

I-Alphon Lipon isidakamizwa esinikeza ukuguquguquka kwezinqubo ze-metabolic.

I-ATX

Ikhodi ye-ATX: A16A X01.

Khipha amafomu nokwakheka

Umuthi lo ukhiqizwa ngendlela yamacwecwe ahlanganiswe ngenhlanganisela ekhethekile yokuvikela. Umthamo ungahluka:

  • I-300 mg - amaphilisi anjalo anomumo we-convex oyindilinga, aphuzi ngombala;
  • I-600 mg - amaphilisi aphuzi aphuzi, anomugqa wokuhlukanisa ezinhlangothini zombili.

Amacwecwe abekwe emabhulokini ezincezu eziyi-10 nezingama-30. Uma kunezingcezu eziyi-10 ku-1 blister, khona-ke amapuleti ama-3 agcwele enqwaba yamakhadibhodi, uma izingcezu ezingama-30, bese kuthi u-1.

Isithako esikhulu somuthi yi-thioctic acid noma i-alpha lipoic acid emthanjeni wama-300 noma ama-600 mg kwithebhulethi eyi-1. Izithako ezingeziwe ezifakiwe ekwakhiweni yilezi: i-cellulose, i-sodium sulfate, i-silicon dioxide, isitashi sommbila, inani elincane le-lactose ne-magnesium stearate.

Isenzo se-Pharmacological

Into esebenzayo iyi-antioxidant yemvelo. Ibandakanya i-decarboxylation yama-alpha-keto acid nge-pyruvic acid. Kulokhu, ukulawulwa kwe-lipid, carbohydrate kanye ne-cholesterol metabolism kwenzeka. Umuthi unezinto eziwohlokayo. Unomphumela omuhle esibindini.

Lapho kukhona isifo sikashukela, ubungozi bokweqisa kwe-lipid peroxidation, okwenzeka ikakhulu ezinhlangeni zepherishi, buyancishiswa. Ngenxa yalokhu, ukujikeleza kwegazi nezinqubo zokushukumisa izinzwa kuyathuthuka. Akunandaba nomphumela we-insulin, into esebenzayo inomthelela ekutholeni kangcono i-glucose emsipha wamathambo.

I-metabolism yomuthi yenzeka esibindini.

I-Pharmacokinetics

Ngemuva kokuphathwa ngomlomo, i-alpha lipoic acid imunwa ngokushesha kusuka emgodini wokugaya ukudla. Metabolism kwenzeka esibindini. Ukuhlushwa okuphezulu kakhulu egazini kuyabonakala emizuzwini embalwa emva kokuthatha iphilisi. Igcotshwe ngokuhlunga kwe-renal ngendlela yama-metabolites amakhulu. Isigamu sempilo sicishe sibe yingxenye yehora.

Yini ebekiwe?

Isibonakaliso esiqondile sokuqokwa kwe-Alpha Lipon ukwelashwa okuphelele kwe-paresthesias ne-polyneuropathy yesifo sikashukela. Umuthi futhi usetshenziselwa i-cirrhosis, i-hepatitis nezinye izilonda zesibindi, ubuthi obuhlukahlukene kanye nokudakwa. Njenge-prophylaxis, ingasetjenziswa njenge-ejenti yokunciphisa i-lipid ye-atherossteosis.

Contraindication

Kunezindlela eziningi zokwephulwa okuqondile kokusetshenziswa kwalesi sidakamizwa. Phakathi kwazo kukhona:

  • ukungabekezelelani kwe-lactose;
  • i-lactose-galactose malabsorption syndrome;
  • ukungasebenzi komongo;
  • ukuthinta nokubeletha;
  • izingane ezingaphansi kweminyaka engu-18;
  • ukungabekezeleli kunoma yiziphi izingxenye zomuthi.
Phakathi kokuphikisana nokusetshenziswa komuthi kukhona izingane ezingaphansi kweminyaka engu-18.
Awukwazi ukusebenzisa umuthi ngesikhathi sokuqunjelwa.
Ukuqwashiswa kuyalulekwa ukuthi uthathe lo muthi nge-pathologies ehlukahlukene yezinso.
Ukuqapha kuyalulekwa ukuthi uthathe lo muthi nge-pathologies yesibindi ehlukahlukene.
Umthamo kufanele ulungiswe kubantu asebekhulile, ngokususelwa kwezinguquko empilweni ejwayelekile yeziguli.

Yonke le mibiko kufanele icatshangwe ngaphambi kokuqala kwenkambo yokwelashwa. Isiguli kufanele sixwayiswe ngazo zonke izingozi ezingaba khona kanye nokuphendula okungahambi kahle.

Ngokunakekela

Ukuqapha kunconyelwa ama-pathologies ahlukahlukene wezinso nesibindi, esimweni se-motor neuropathy. Umthamo kufanele ulungiswe kubantu asebekhulile, ngokususelwa kwezinguquko empilweni ejwayelekile yeziguli.

Ungayithatha kanjani i-Alfa Lipon?

Kungcono ukuphuza amaphilisi imizuzu engama-30 ngaphambi kokudla okuyinhloko. Uma uphuza amaphilisi ngokudla, khona-ke ukumunyiswa kwento esebenzayo yehlisa ijubane futhi umphumela wokwelapha awutholakalanga masinyane. Inkambo yokwelashwa iphindwa kabili ngonyaka.

Ngokuthuthukiswa kwe-polyneuropathy ekuqaleni kokwelashwa, kunconywa ukuphatha kwabazali umuthi. Umthamo wokuqala wansuku zonke unqunyelwe i-600-900 mg ngaphakathi. Umuthi uyancibilika kwisixazululo se-isotonic sodium chloride. Izifundo ezinjalo zokwelashwa zihlala okungenani amaviki ama-2. Ezimweni ezibucayi kakhulu, umthamo unyuka ufike kuma-1200 mg ngosuku. Ukwelashwa kwesondlo kungama-600 mg ngosuku, ahlukaniswe ngemithamo emithathu. Ukwelashwa okunjalo kungahlala izinyanga ezi-3.

Ngoshukela

Ekwelapheni i-neuropathy yesifo sikashukela, umthamo wokuqala wansuku zonke ungama-300 mg ngokuqondile noma ama-200 mg kathathu ngosuku izinsuku ezingama-20. Ngemuva kwalokho thatha umthamo wokulungisa inani elingama-400-600 mg wezinyanga ezi-1-2. Indlela eyengeziwe ukusetshenziswa kwezidakamizwa zomlomo ze-hypoglycemic.

Ekwelapheni i-neuropathy yesifo sikashukela, umthamo wokuqala wansuku zonke ungama-300 mg ngokuqondile noma ama-200 mg kathathu ngosuku izinsuku ezingama-20.

Ukwehla kwesisindo

Ukuze ulahlekelwe isisindo, kunconywa ukuphuza i-tablet izikhathi ezi-2 ngosuku. Kepha iziguli kufanele ziqonde ukuthi amanye amaphilisi awakwazi ukufaka isandla ekwehliseni isisindo nokugcinwa. Amane ayingxenye yokwelashwa okuyinkimbinkimbi. Okuphoqelekile kuleli cala kuzoba ukuvivinya umzimba okulinganiselayo kanye nokubambelela ngokuqinile ekudleni.

Imiphumela emibi ye-Alfa Lipon

Ngomthamo ofanele, imiphumela emibi ayivelakakhulu. Ngokuyisisekelo, aboniswa ukuncipha kweglucose yegazi, okubonisa ukukhula kwe-hypoglycemia. Lesi simo sihambisana nokuqaqanjelwa yikhanda nesiyezi, ukuncipha okubukwayo nokuqina kokujuluka.

Imvamisa, ipheshana lesisu liphendula umuthi. Isiguli singabuzwa ubuhlungu besisu, isicanucanu nokuhlanza, isifo sohudo. Mhlawumbe ukubonakala kokuqubuka kwesikhumba, kuhambisane nokulunywa, nokukhula kwe-eczema.

Umthelela ekhonweni lokulawula izindlela

Ngenxa yengozi ephezulu ye-hypoglycemia, isiyezi esinokwenzeka kanye nombono onciphile, kunconyelwa ukuba uqaphele ngesikhathi sokwelashwa futhi unciphise ukuphathwa kwezimoto nezinye izindlela eziyinkimbinkimbi ezidinga ukunakwa okwandayo kokunakwa.

Imiyalo ekhethekile

Ngakuqala kokwelashwa, kunganda ukubekeka engcupheni ye-paresthesia, okumele ibhekwe lapho kwenziwa ukwelashwa. Ngenxa yokuvuswa kwezinqubo zokuvuselela kabusha, iziguli zingaba nezimpukane phambi kwamehlo abo.

Isifo sohudo singenye yemiphumela emibi yokuphuza umuthi.

Kuyadingeka ukubheka njalo izinkomba ze-glucose yabantu abanesifo sikashukela esitholakele. Ukuze uvimbele ukukhula kwe-hypoglycemia, unganciphisa umthamo womuthi uma usetshenziswa njenge-ejenti ye-antidiabetesic.

Udayi, oyingxenye yegobolondo lethebhulethi, angavusa ukuthuthukiswa kokubonakala komzimba.

Sebenzisa ebudaleni

Kwabadala, kuthathwa umthamo wansuku zonke osezingeni elifanele. Umthamo uguqulwa ucatshangelwa izinguquko ezimweni ezijwayelekile zempilo zesiguli.

Ukunquma i-Alpha Lipon Yezingane

Leli thuluzi alisetshenziswa emisebenzini yezingane.

Sebenzisa ngesikhathi sokukhulelwa nokukhishwa komzimba

Akunconyelwe ukuphuza amaphilisi ngesikhathi sokukhulelwa. Ngoba akukho datha ethembekile yokuthi ingabe into esebenzayo inomphumela ongemuhle ku-fetus, ukwelashwa okunjalo kuyinto engathandeki.

Isikhathi sokulashwa kwezidakamizwa, kungcono ukwenqaba ukuncelisa ibele.

Akunconyelwe ukuphuza amaphilisi ngesikhathi sokukhulelwa.

Isicelo sokusebenza kokulimala kwezinso

Umthamo kuleli cala uzoncika ekuthini imvume ye-creatinine. Uma iphansi, yehlisa umthamo womuthi obekelwe isiguli. Uma ukuhlolwa kushintsha kube kubi, kungcono ukuyeka ukwelashwa okunjalo.

Isicelo sokusebenza kokulimala kwesibindi

Ngama-pathologies wesibindi, umuthi uthathwa ngokunakekelwa okukhulu. Ekuqaleni, kuthathwa umthamo omncane wesidakamizwa. Uma ukuhlolwa kokuqina kwesibindi kuya ngokuya kukhula, ukwelashwa kuyamiswa.

Ukweqisa kwe-Alfa Lipon

Azikho izimpawu ezinzima ze-overdose eziqaphelekayo. Kodwa izimpawu zokuphendula okungahambi kahle zinganda.

Ukuxhumana nezinye izidakamizwa

Umuthi unciphisa ukusebenza kweCisplatin. Umuthi awuthathwa ngemikhiqizo yobisi kanye nosawoti wensimbi. Ungathathi noma yiziphi izithasiselo zokudla okunempilo eziqukethe inani elikhulu le-iron ne-magnesium.

Umuthi unciphisa ukusebenza kweCisplatin.

I-Thioctic acid ikhulisa imiphumela yezidakamizwa ezinciphisa ushukela ngomlomo, ezinye izidakamizwa zokulwa nesifo sikashukela ezigulini ezinesifo sikashukela.

Ama-antioxidants athuthukisa umphumela we-antidiabetesic wezidakamizwa. Kuyadingeka ukubheka njalo izinga le-lactose egazini, ngoba into esebenzayo ingakushintsha kakhulu ukuqina kwayo. Lokhu kuyiqiniso ikakhulukazi kwiziguli ezinokuntuleka kwe-enzyme lactase.

Ukuhambisana notshwala

Awukwazi ukuhlanganisa ukuphuza kwamathebulethi nokuphuza utshwala, njengoba lokhu kuthuthukisa ukungasebenzi kahle komuthi kanye nokwehla komphumela wawo wokwelapha. Izimpawu zokudakwa zizoqina, ezithinta kabi isimo somzimba.

Ama-Analog

Kunokufana okuningana kwalo muthi okufana nakho ngokuya ngezinto ezisebenzayo kanye nomphumela wokwelapha. Abaziwa kakhulu kubo:

  • I-Berlition;
  • I-Dialipon;
  • Tio Lipon;
  • U-Espa Lipon;
  • I-Thiogma;
  • I-Thioctodar.

Ukukhetha kokugcina kwezidakamizwa kuhlala nodokotela ohambelayo.

I-Alpha Lipoic Acid yesifo sikashukela se-Neuropathy

Imibandela yekhefu lekhemisi

Ungayithenga cishe kunoma iyiphi ikhemisi ngomuthi onikezwe.

Ngingakwazi ukuthenga ngaphandle kadokotela?

Umuthi uhanjiswa emaphoyiseni asekhemisi kuphela uma kunikezwa incwadi kadokotela ekhethekile evela kudokotela.

Intengo ye-Alfa Lipon

Intengo yomuthi enomthamo we-300 mg cishe ngama-ruble angama-320. ngephakeji ngalinye, nangomthamo wama-ruble angama-600 - ama-ruble angama-550.

Izimo zokugcina zomuthi

Endaweni eyomile nebumnyama, emazingeni okushisa asekamelweni, lapho izingane zingafinyeleleki khona.

Isikhathi sokuphelelwa yisikhathi

Hhayi iminyaka engaphezu kwemi-2 kusuka ngosuku lokukhipha olukhonjiswe kwiphakheji yangempela.

Umkhiqizi

Inkampani yezokukhiqiza: I-PJSC "I-Kiev Vitamin Plant". EKiev, e-Ukraine.

Umuthi uhanjiswa emaphoyiseni asekhemisi kuphela uma kunikezwa incwadi kadokotela ekhethekile evela kudokotela.

Ukubuyekezwa ku-Alfa Lipon

UVictor, oneminyaka engama-37

Umuthi muhle. Yachazwa ngemuva kobuthi botshwala. Kusebenze kahle njenge-ejenti yokwehlisa umoya. Okubi kuphela ukuthi udinga ukuphuza amaphilisi isikhathi eside, kusukela ezinyangeni ezi-1 kuye kwezi-3. Ngoba ubuthi babunzima kakhulu, ngabe sengiyithatha izinyanga ezintathu.

U-Elena, oneminyaka engama-43 ubudala

I-Lipoic acid yabekwa njenge-hepatoprotector lapho nginezinkinga ezinzima zesibindi. Umuthi waphuzwa kakhulu njengokuyalelwa udokotela owayeyinyanga eyodwa, futhi wasiza. Hhayi isimo sesibindi kuphela, kepha namanye amalungu angaphakathi athuthukisiwe. Ngijabule ngomuthi. Okuwukuphela kokubi ukuthi ayikho kuwo wonke amakhambi emithi.

UMikhail, oneminyaka engama-56

Sekuphele iminyaka ngihlaselwa isifo sikashukela. Inkambo ene-Alfa Lipon ichazwe njengokwelashwa kokulungiswa. Anginazikhalazo ngaye. Akubangeli lutho olubi lokuphendula, futhi intengo inengqondo. Ngiweluleka lo muthi.

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