Umuthi i-Emoxipin Plus: imiyalo esetshenzisiwe

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I-Emoxipin Plus iyi-angioprotector, etholakala ngesimo sezisombululo futhi isetshenziswa ekwelapheni nasekuvimbeleni izifo zamehlo. Ngokusebenzisa njalo i-antioxidant, ukwehla kokuqina kwemithambo nokuthuthuka kwe-microcirculation yegazi kuyabonakala. Ukwethulwa kwezixazululo zomjovo kwenziwa ngezindlela eziningana, kufaka phakathi i-intramuscular and intravenous. Kuyathengiswa kunamaconsi wamehlo wegama elifanayo. Contraindication kanye nemiphumela emibi yemithi emzimbeni wesiguli ichaziwe emiyalweni.

Igama Lezwe elingafanele

Iqembu negama lamanye amazwe yiMethylethylpyridinol, ngesiLatini - Methylethylpiridinol.

I-Emoxipin Plus iyi-angioprotector, etholakala ngesimo sezisombululo futhi isetshenziswa ekwelapheni nasekuvimbeleni izifo zamehlo.

I-ATX

Ikhodi eyodwa ye-ATX yemithi yi-C05CX (iphelelwe yisikhathi - S01XA).

Khipha amafomu nokwakheka

Umuthi uyatholakala ngesimo soketshezi. Izinhlobo eziphambili zokukhishwa zifaka:

  • ukumiswa kokuphathwa kwe-i / m (intramuscularly) kanye ne-iv (intravenously);
  • iso lihla.

Umenzi unikeza into eyodwa esebenzayo kuwo wonke amafomu umthamo - methylethylpyridinol hydrochloride. Ukuqoqwa kwento esemqoka kuyahluka ngokuya ngohlobo lokukhululwa. Izici ezisizayo zikhona.

Amaconsi

I-eye yehla ngokubukeka - u-opalescent omncane, uketshezi olunombala noma olunemibala kancane ngaphandle kwephunga elithile. Isixazululo sithengiswa emabhodleleni engilazi amnyama afakwe i-dispenser cap. Umthamo wesitsha ngu-5 ml.

Okuqukethwe kwesakhi esiyinhloko yi-10 mg. Izakhi ezingeziwe ekwakhiweni kwefomu lomthamo:

  • amanzi ahlanziwe;
  • i-sodium benzoate;
  • potassium dihydrogen phosphate;
  • sodium hydrogen phosphate dodecahydrate;
  • i-anhydrous sodium sulfite;
  • i-soluble methyl cellulose.

Izindlwana ezine-dispenser zifakwe emabhokisini amakhadibhodi ngenani le-1 pc. Ngaphezu kwesitsha, iphakethe liqukethe imiyalo esetshenzisiwe.

I-Emoxipin itholakala njengamaconsi eso.

Isixazululo

Ukumiswa koketshezi olungenamibala, akuvamile ukuba lube ophuzi ngenani elincane lezinhlayiya eziqinile. Ukuxakaniseka kwento esebenzayo ayidluli kuma-30 mg. Uhlu lwezinto ezisizayo:

  • amanzi ahlanziwe;
  • sodium hydroxide (isixazululo).

Isixazululo sithululelwa kuma-ampoules engilazi ecwengekile ngevolumu engu-1 ml noma i-5 ml. Amaphakeji aqukethe amaselula aqukethe ama-ampoules ayi-5. Emaphepheni amakhadibhodi kukhona amaphakheji we-1, 5, 10, 20, 50 noma we-100. Kuyathengiswa ikhambi lomjovo (intramuscular).

Uhlobo olungekho

Umuthi awutholakali ngohlobo lwamafutha okugcoba, amaphilisi, amaphilisi kanye nemisele.

Isenzo se-Pharmacological

Imiphumela yokwelashwa yikhono lomuthi lokukhipha i-angioprotective, antioxidant, antihypoxic effect emzimbeni. Into esemqoka inciphisa ukuqina kwamadonga we-capillary, ukuhlanganiswa kweplatelet. Isebenza njenge-inhibitor ekhethiwe yezinqubo zokukhulula zamahhala.

Ubungozi bokukhubazeka kanye nokusetshenziswa okuhleliwe komuthi buncishisiwe. Ngama-pathologies wezinhliziyo nemizwa, umuthi wehlisa ubudisi kanye nobukhulu bezimpawu ezihambisana nalesi sifo. Kulokhu, kukhona ukwanda kokumelana kwezicubu ze-ischemia ne-hypoxia.

Izixazululo zokuphathwa kwe-intravenous kanye ne-intramuscular ngcono ukuqina nokusebenza okuvumayo kohlelo lwethambo nenhliziyo. Ngokusetshenziswa isikhathi eside kwekhambi lomjovo, ukwehla kokugxila kwe-tisc necrosis kubonwa nge-myocardial infarction. Ukwanda kwemikhumbi ye-coronary kungenxa yekhono lomuthi lokuba nomthelela we-hypotensive emzimbeni.

Umphumela we-retinoprotective we-antioxidant uvikela i-retina kusuka ekukhuthazeleni kwangaphandle, kufaka phakathi imithombo yokukhanya yokufakelwa. Amaconsi eshesha asheshisa ukubuyiselwa kwamathambo we-hemorrhages angabanzi kakhulu. Ngokusebenzisa okuhleliwe, ulwelwesi lwamaseli luyavuselelwa futhi nezindonga zemithambo ziba ngaphezulu.

Umuthi i-Emoksipin uvikela i-retina ethonyeni lokuthonya langaphandle.

I-Pharmacokinetics

Izinto ezisebenzayo zidonswa ngokushesha zingene egazini futhi zifinyelele izicubu ezithintekile, kungakhathalekile ukuthi iyiphi indlela yokuphatha. Ukuhlaziywa okukhulu nge-iv nokuphathwa kwe-intramuscular kutholakala imizuzu eyi-15 ngemuva komthamo wokuqala. I-Metabolism yenziwa isibindi, ama-metabolites angasebenzi akhiqizwa inqubo. Ukuhlanganiswa kwamaprotheni egazi - hhayi ngaphezu kwama-54%. Kushiya umzimba ngomchamo. Isikhathi sokuqothula yimizuzu engama-30 ukuya kwengama-35.

Amaconsi wamehlo angama-40% aboshelwe kumaprotheni egazi. Iqoqelalwazi eliphezulu le-element main izicubu liphakeme kunakwigazi le-plasma. Ama-Metabolites (imikhiqizo ehlanganisiwe kanye ne-desalkylated) adalulwa yizinso.

Okunqunyelwe

Umuthi usetshenziselwa i-cardiology, ophthalmology, neurosurgery ne-neurology. Kusetshenziswa isixazululo se-i / m kanye nokuphathwa kwe-iv lapho kutholwa ama-pathologies alandelayo esigulini:

  • ischemic stroke;
  • i-hemorrhagic stroke (ngesikhathi sokuvuselelwa);
  • ingozi ye-cerebrovascular;
  • infarction myocardial;
  • i-angina pectoris engazinzi;
  • i-reperfusion syndrome (ukuvimbela);
  • I-TBI (ukulimala kobuchopho obuxakayo);
  • intracerebral, hemmatoma and subdural hematomas.

Izinkomba ezisetshenziselwa amaconsi wamehlo:

  • ama-hemorrhages egumbini elingaphandle le-ophthalmic;
  • Izinkinga ze-myopia;
  • glaucoma
  • ikati
  • i-retinopathy
  • ukushiswa kanye nokuvuvukala komqubuko.

Amaconsi wamehlo angasetjenziswa ekwelapheni ama-hemorrhages ku-sclera.

I-Emoxipin yezidakamizwa isetshenziselwa ukuphazamiseka kwe-cerebrovascular.
I-Emoxipin yezidakamizwa isetshenziselwa ukufakwa kwe-myocardial infarction.
I-Emoxipin yezidakamizwa isetshenziselwa izinkinga ze-myopia.

Contraindication

Ukusetshenziswa kwanoma yiluphi uhlobo lomthamo akunakwenzeka uma isiguli sine-contraindication. Lokhu kufaka phakathi:

  • i-trimester yokugcina yokukhulelwa;
  • inkathi yokuhlanza;
  • iminyaka yezingane (kuze kube iminyaka eyi-18);
  • ukungabekezelelani ngakunye ezintweni eziyinhloko noma ezisizayo.

Ukuqapha kunconywa kwiziguli esezikhulile nabantu abane-pathologies yesibindi.

Ungayithatha kanjani i-Emoxipin Plus

Ukwethulwa kwekhambi ku / m kanye / ku kwenziwa nge-Drip. Ilungiselelwe ngokushesha ngaphambi kwenqubo emizuzwini engama-5-7. Umthamo ophakanyisiwe wokwelapha kufanele uchitheke ku-isotonic sodium chloride. Umthamo unqunywa ngawodwana. Imiyalo ikhombisa uhlobo lokulinganiselwa lwesilinganiso:

  • phakathi naphakathi - 10 mg / kg yesisindo 1 isikhathi ngosuku;
  • intramuscularly - akukho ngaphezu kwama-60 mg kanye izikhathi ezingama-2-3 ngosuku.

Isikhathi sokusetshenziswa siyizinsuku eziyi-10-30. Ukuthola imiphumela ephezulu, kunconyelwa ukuphatha isixazululo ngaphakathi kwezinsuku ezingama-5-8, sonke isikhathi, ukuphatha umuthi nge-intramuscularly.

I-Emoxipin yezidakamizwa iyatholakala kuma-ampoules.

Ukufakwa kwamaconsi kwenziwa ku-conjunctival sac. Ngaphambi kwenqubo, kuyadingeka ukuvula ibhodlela, gqoka i-dispenser futhi unikine ngamandla. Isitsha siphendulwe sabheka phansi. Ukucindezela i-dispenser kuzokwenza kube lula ukubala inani elidingekayo lamaconsi. Isimo sokwelapha isiguli esikhulile sihla kathathu ngosuku. Inkambo yokwelashwa ezimweni eziningi yizinsuku ezingama-30. Uma kunesidingo, inganwetshwa ize ifinyelele ezinsukwini ezingama-180.

Ngoshukela

Iziguli ezinesifo sikashukela zingadinga ukulungiswa komthamo. Ukwelashwa kufanele kuqalwe ngomthamo wesigamu.

Imiphumela emibi ye-Emoxipin Plus

Umuthi onokulawulwa okungafanele noma obedlula okujwayelekile ukwelashwa ucasisa ukuthuthukiswa kwemiphumela emibi evela ohlelweni lwezinzwa oluphakathi nezitho zangaphakathi. Lokhu kufaka phakathi:

  • izinzwa zobuhlungu kanye nokuvutha kwemizwa endaweni yomjovo;
  • ukozela
  • ukweqile;
  • isifo se-metabolic (akuvamile);
  • ukwanda kwengcindezi yegazi;
  • ukukhuphuka kwenhliziyo;
  • i-migraine
  • umuzwa ovuthayo emehlweni;
  • ukulunywa
  • hyperemia.

Ukungezwani komzimba kubonwa kuma-26% eziguli. Zibonakala njengokubomvu esikhunjeni, emaphashini nasekuwuncineni.

Imiphumela emibi ye-Emoxipin ibonakaliswa ubuthongo.
Umphumela omubi we-Emoxipin ukwanda komfutho wegazi.
Umphumela omubi we-Emoxipin ukwanda kwenhliziyo.
Umphumela omubi we-Emoxipin yi-migraine.
Imiphumela emibi ye-Emoxipin ibonakaliswa umuzwa ovuthayo emehlweni.
Imiphumela emibi ye-Emoxipin ibonakaliswa ngendlela yokulunywa.

Imiyalo ekhethekile

Ukuphathwa kwe-Intravenous kudinga ukuqapha ngokucophelela umfutho wegazi nokuqunjelwa kwegazi. Ngokusebenzisa kanye kanyekanye amaconsi wamehlo kubakhiqizi abahlukahlukene, ukufakwa kwe-angioprotector kunconyelwe ukwenziwa ekugcineni. Isikhathi sokuphakathi kokufakwa kufanele sibe imizuzu engama-20-25.

Ngesikhathi sokuqhaqhazela, amafomu amagwebu, angathinti ikhwalithi yomuthi. Foam inyamalala ngokwayo ngemuva kwemizuzwana eyi-15-30. Ukusetshenziswa isikhathi eside kwesidakamizwa kuthinta izinga le-lycopene (antioxidant, i-carotenoid pigment) emzimbeni.

Sebenzisa ebudaleni

Ezigulini esezikhulile, kungcono ukusebenzisa umjovo we-intramuscular ukugwema ukwakheka kwe-hematomas. Kunconywe ukusetshenziswa kwengxenye yemithamo.

Ukunquma i-Emoxipin Plus ezinganeni

Imithi (kungakhathalekile ukuthi ifomu lomthamo) ayinqunyelwe iziguli ezingaphansi kweminyaka engu-18.

Sebenzisa ngesikhathi sokukhulelwa nokukhishwa komzimba

Ukusetshenziswa kwesidakamizwa ngesikhathi sokukhulelwa nokuzala ingane akuvunyelwe ngokuphelele.

Ukweqisa kwe-Emoxipin Plus

Amacala okweqa ngokweqile ayivelakancane. Zihambisana nezimpawu zobuntu, kufaka phakathi isicanucanu, ukuhlanza, izinhlungu esiswini. Ukwelashwa okubonakalayo, ukuphathwa kwama-enterosorbents kanye ne-gastric lavage kuyadingeka.

Umuthi i-Emoxipin (kungakhathalekile ukuthi ifomu lomthamo) awunqunyelwe ezigulini ezingaphansi kweminyaka engu-18.

Ukuxhumana nezinye izidakamizwa

Izisombululo ze-infusion azikhuthazwanga ukuthi zisetshenziswe kanyekanye namanye amalungiselelo we-vascular, ama-antibiotics kanye ne-proton pump inhibitors. Izidakamizwa ezingenhla zinganciphisa umsebenzi kanye ne-bioavailability ye-angioprotector. Ukusetshenziswa kanyekanye kwezidakamizwa nezidakamizwa ezingama-antiviral kukhuthaza ukukhula kokuhluleka kwesibindi ngenxa yomthwalo omkhulu kulesi sitho.

Amaconsi wamehlo angahlanganiswa nemithi ye-herbal (i-ginkgo biloba ekhishwe, i-blueberries) ethuthukisa umbono. Ukusetshenziswa kwamaconsi kungahambisana nemijovo ye-intramuscular of amavithamini.

Ukuhambisana notshwala

Umuthi awuhambelani ne-ethanol. Ukusetshenziswa kotshwala ngesikhathi sokwelashwa kwenqatshelwe ngokuphelele.

Ama-Analog

I-angioprotector inezindawo eziningi ezinomphumela ofanayo wokwelapha. Abalingani abaningi abenziwe ngaphakathi basendleleni ephakathi yamanani futhi bayatholakala kwiziguli eziningi. Lokhu kufaka phakathi:

  1. I-Emoxipin-Akti. Analogue yesakhiwo yoqobo. Into efanayo esebenzayo ekuqoqweni okuncane inomphumela we-angioprotective ne-antioxidant emzimbeni wesiguli. Ukusetshenziswa ngezinjongo zokuvimbela nokwelapha kuvunyelwe ku-ophthalmology, inhliziyo and neurosurgery. Kukhona ukuphambana. Intengo emakhemisi isuka kuma-ruble angama-200.
  2. Isazi se-Emoxy. Kutholakala ngesimo samaconsi e-ophthalmic. Isetjenziswa ngaphezulu ngezinhloso zokwelapha kuphela ezigulini ezindala. Ukwakheka kuqukethe i-methylethylpyridinol hydrochloride (10 mg). Mhlawumbe ukuthuthukiswa kwemiphumela emibi. Izindleko - kusuka kuma-ruble angama-90.
  3. I-Cardioxypine. I-angioprotector enamandla esisiza ukunciphisa ukuncipha kwemithambo yegazi. Ngokusetshenziswa njalo, izitsha zobuchopho ziba namandla ngokwengeziwe kwi-hypoxia. Ukusetshenziswa ngezinjongo zokwelapha kanye ne-prophylactic kwenziwa ngemvume kadokotela. Intengo - kusuka kuma-ruble angama-250.
  4. Methylethylpyridinol-Eskom. Analogue yezakhiwo zesidakamizwa sokuqala. Ukuqanjwa kufana ngokuphelele, njengoba kunjalo izinkomba zokusetshenziswa. Imiphumela emibi nokuphikisana okuphelele kubekwe kwimiyalo. Izindleko emakhemisi zivela kuma-ruble ayi-143.

Ukukhethwa komuntu obambele esikhundleni kwenziwa ngudokotela oholayo uma isiguli sinokuphikisana ngokuphelele nokusetshenziswa komuthi ngenhloso yokuvimbela nokwelapha.

Ividiyo yokuqeqeshwa ye-Emoxipin
Amaconsi e-glaucoma: IBetaxolol, iTravatan, iTaurine, iTaufon, i-Emoxipine, iQuinax, iCatachrome
I-Ophthalmologist mayelana ne-HARM DROP ne-EYES / Dry eye syndrome ebomvu
I-Conjunctivitis. Yini eyenza amehlo ami aqhume

Imibandela yekhefu lekhemisi

Dinga umuthi weholide emakhemisi.

Ngingakwazi ukuthenga ngaphandle kadokotela

Umuthi awunakuthengwa ngaphandle kwencwadi kadokotela ekhethekile.

Intengo ye-Emoxipin Plus

Izindleko zomuthi emakhemisi zivela kuma-ruble ayi-135.

Izimo zokugcina zomuthi

Indawo yokubeka kufanele ibe yinhle futhi ibe mnyama, ingafinyeleleki ezinganeni nasezilwaneni.

Isikhathi sokuphelelwa yisikhathi

Impilo yeshalofu yesisombululo yizinyanga ezingama-36, amaconsi e-ophthalmic - azidluli izinyanga ezingama-24.

I-Cardioxypine iyi-analogue ye-Emoxipin yokulungiselela.

Umkhiqizi

I-Enzyme (Russia), Tallinn Pharmaceutical Plant (Estonia).

Ukubuyekezwa kwe-Emoxipin Plus

U-Evgenia Bogorodova, udokotela wezifo zenhliziyo, iYekaterinburg

Lapho ngisebenza, ngisebenzisa lo muthi isikhathi esingaphezu kweminyaka emi-5. Nginikeza iziguli ezimweni ezimbi kakhulu, zinamandla. I-Angioprotector ithuthukisa i-microcirculation yegazi futhi inomphumela onenzuzo ebuchosheni. Ngokusebenzisa njalo, ubungozi bokuhlaselwa yisifo senhliziyo nemivimbo kuncishiswa kaningana. Ngaphezu kwalokho, umuthi uvikela ubuchopho ekubulaleni i-oksijini.

Imiphumela emibi yenzeka ezigulini eziningi ngenxa yezimpawu zomzimba ngamunye. Imvamisa kakhulu le yimiphumela yokungezwani komzimba (i-acne, redness yezingqimba ezingehla ze-dermis) ne-dyspepsia Isiguli siba nobuhlungu be-epigastric, isicanucanu, nokuhlanza. Ukwelashwa okubonakalayo kufanele kukhethwe ngokucophelela, awukwazi ukukhetha umuthi ngokwakho.

U-Elena, oneminyaka engama-46, eSt

Ngezokwelapha ngasebenzisa amaconsi e-ophthalmic. IGlaucoma yatholakala eminyakeni eminingana eyedlule, futhi yelashwa isikhathi eside. Imithambo yegazi ibe buthaka, waqala wabona ukuthi ama-capillaries ahlala eqhuma. Ama-hematomas kwabamhlophe bamehlo anyamalala isikhathi eside, amaconsi ajwayelekile awazange asize okuningi. Ngenxa yalokhu, umbono wawela, iso elilodwa laba nzima ukubona. Ngaphendukela ku-ophthalmologist ukuthola izeluleko, weluleka i-angioprotector eyenziwe ekhaya.

Ngathenga umuthi onikezwe umuthi. Kusetshenziswe ngokwemiyalo - kudonsa kabili kanye esweni ngalinye kabili ngosuku. Imiphumela emibi yavela ngosuku lokuqala. Amehlo akhe ayeshayekile futhi enamanzi. Kwavela amabala abomvu ezinqeni. Ngangesaba ukusebenzisa amafutha e-antihistamine, ngathambisa izinkophe ngo-ukhilimu wengane. Naphezu kokwenqatshwa, umuthi wasiza ngokushesha. I-hematoma ixazululwe ngokuphelele ezinsukwini ezi-2, umbono wabuyiselwa ngokuphelele ngemuva kwezinsuku ezingama-4.

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