I-Emoxipin Plus iyi-angioprotector, etholakala ngesimo sezisombululo futhi isetshenziswa ekwelapheni nasekuvimbeleni izifo zamehlo. Ngokusebenzisa njalo i-antioxidant, ukwehla kokuqina kwemithambo nokuthuthuka kwe-microcirculation yegazi kuyabonakala. Ukwethulwa kwezixazululo zomjovo kwenziwa ngezindlela eziningana, kufaka phakathi i-intramuscular and intravenous. Kuyathengiswa kunamaconsi wamehlo wegama elifanayo. Contraindication kanye nemiphumela emibi yemithi emzimbeni wesiguli ichaziwe emiyalweni.
Igama Lezwe elingafanele
Iqembu negama lamanye amazwe yiMethylethylpyridinol, ngesiLatini - Methylethylpiridinol.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu.jpg)
I-Emoxipin Plus iyi-angioprotector, etholakala ngesimo sezisombululo futhi isetshenziswa ekwelapheni nasekuvimbeleni izifo zamehlo.
I-ATX
Ikhodi eyodwa ye-ATX yemithi yi-C05CX (iphelelwe yisikhathi - S01XA).
Khipha amafomu nokwakheka
Umuthi uyatholakala ngesimo soketshezi. Izinhlobo eziphambili zokukhishwa zifaka:
- ukumiswa kokuphathwa kwe-i / m (intramuscularly) kanye ne-iv (intravenously);
- iso lihla.
Umenzi unikeza into eyodwa esebenzayo kuwo wonke amafomu umthamo - methylethylpyridinol hydrochloride. Ukuqoqwa kwento esemqoka kuyahluka ngokuya ngohlobo lokukhululwa. Izici ezisizayo zikhona.
Amaconsi
I-eye yehla ngokubukeka - u-opalescent omncane, uketshezi olunombala noma olunemibala kancane ngaphandle kwephunga elithile. Isixazululo sithengiswa emabhodleleni engilazi amnyama afakwe i-dispenser cap. Umthamo wesitsha ngu-5 ml.
Okuqukethwe kwesakhi esiyinhloko yi-10 mg. Izakhi ezingeziwe ekwakhiweni kwefomu lomthamo:
- amanzi ahlanziwe;
- i-sodium benzoate;
- potassium dihydrogen phosphate;
- sodium hydrogen phosphate dodecahydrate;
- i-anhydrous sodium sulfite;
- i-soluble methyl cellulose.
Izindlwana ezine-dispenser zifakwe emabhokisini amakhadibhodi ngenani le-1 pc. Ngaphezu kwesitsha, iphakethe liqukethe imiyalo esetshenzisiwe.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-2.jpg)
I-Emoxipin itholakala njengamaconsi eso.
Isixazululo
Ukumiswa koketshezi olungenamibala, akuvamile ukuba lube ophuzi ngenani elincane lezinhlayiya eziqinile. Ukuxakaniseka kwento esebenzayo ayidluli kuma-30 mg. Uhlu lwezinto ezisizayo:
- amanzi ahlanziwe;
- sodium hydroxide (isixazululo).
Isixazululo sithululelwa kuma-ampoules engilazi ecwengekile ngevolumu engu-1 ml noma i-5 ml. Amaphakeji aqukethe amaselula aqukethe ama-ampoules ayi-5. Emaphepheni amakhadibhodi kukhona amaphakheji we-1, 5, 10, 20, 50 noma we-100. Kuyathengiswa ikhambi lomjovo (intramuscular).
Uhlobo olungekho
Umuthi awutholakali ngohlobo lwamafutha okugcoba, amaphilisi, amaphilisi kanye nemisele.
Isenzo se-Pharmacological
Imiphumela yokwelashwa yikhono lomuthi lokukhipha i-angioprotective, antioxidant, antihypoxic effect emzimbeni. Into esemqoka inciphisa ukuqina kwamadonga we-capillary, ukuhlanganiswa kweplatelet. Isebenza njenge-inhibitor ekhethiwe yezinqubo zokukhulula zamahhala.
Ubungozi bokukhubazeka kanye nokusetshenziswa okuhleliwe komuthi buncishisiwe. Ngama-pathologies wezinhliziyo nemizwa, umuthi wehlisa ubudisi kanye nobukhulu bezimpawu ezihambisana nalesi sifo. Kulokhu, kukhona ukwanda kokumelana kwezicubu ze-ischemia ne-hypoxia.
Izixazululo zokuphathwa kwe-intravenous kanye ne-intramuscular ngcono ukuqina nokusebenza okuvumayo kohlelo lwethambo nenhliziyo. Ngokusetshenziswa isikhathi eside kwekhambi lomjovo, ukwehla kokugxila kwe-tisc necrosis kubonwa nge-myocardial infarction. Ukwanda kwemikhumbi ye-coronary kungenxa yekhono lomuthi lokuba nomthelela we-hypotensive emzimbeni.
Umphumela we-retinoprotective we-antioxidant uvikela i-retina kusuka ekukhuthazeleni kwangaphandle, kufaka phakathi imithombo yokukhanya yokufakelwa. Amaconsi eshesha asheshisa ukubuyiselwa kwamathambo we-hemorrhages angabanzi kakhulu. Ngokusebenzisa okuhleliwe, ulwelwesi lwamaseli luyavuselelwa futhi nezindonga zemithambo ziba ngaphezulu.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-3.jpg)
Umuthi i-Emoksipin uvikela i-retina ethonyeni lokuthonya langaphandle.
I-Pharmacokinetics
Izinto ezisebenzayo zidonswa ngokushesha zingene egazini futhi zifinyelele izicubu ezithintekile, kungakhathalekile ukuthi iyiphi indlela yokuphatha. Ukuhlaziywa okukhulu nge-iv nokuphathwa kwe-intramuscular kutholakala imizuzu eyi-15 ngemuva komthamo wokuqala. I-Metabolism yenziwa isibindi, ama-metabolites angasebenzi akhiqizwa inqubo. Ukuhlanganiswa kwamaprotheni egazi - hhayi ngaphezu kwama-54%. Kushiya umzimba ngomchamo. Isikhathi sokuqothula yimizuzu engama-30 ukuya kwengama-35.
Amaconsi wamehlo angama-40% aboshelwe kumaprotheni egazi. Iqoqelalwazi eliphezulu le-element main izicubu liphakeme kunakwigazi le-plasma. Ama-Metabolites (imikhiqizo ehlanganisiwe kanye ne-desalkylated) adalulwa yizinso.
Okunqunyelwe
Umuthi usetshenziselwa i-cardiology, ophthalmology, neurosurgery ne-neurology. Kusetshenziswa isixazululo se-i / m kanye nokuphathwa kwe-iv lapho kutholwa ama-pathologies alandelayo esigulini:
- ischemic stroke;
- i-hemorrhagic stroke (ngesikhathi sokuvuselelwa);
- ingozi ye-cerebrovascular;
- infarction myocardial;
- i-angina pectoris engazinzi;
- i-reperfusion syndrome (ukuvimbela);
- I-TBI (ukulimala kobuchopho obuxakayo);
- intracerebral, hemmatoma and subdural hematomas.
Izinkomba ezisetshenziselwa amaconsi wamehlo:
- ama-hemorrhages egumbini elingaphandle le-ophthalmic;
- Izinkinga ze-myopia;
- glaucoma
- ikati
- i-retinopathy
- ukushiswa kanye nokuvuvukala komqubuko.
Amaconsi wamehlo angasetjenziswa ekwelapheni ama-hemorrhages ku-sclera.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-4.jpg)
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Contraindication
Ukusetshenziswa kwanoma yiluphi uhlobo lomthamo akunakwenzeka uma isiguli sine-contraindication. Lokhu kufaka phakathi:
- i-trimester yokugcina yokukhulelwa;
- inkathi yokuhlanza;
- iminyaka yezingane (kuze kube iminyaka eyi-18);
- ukungabekezelelani ngakunye ezintweni eziyinhloko noma ezisizayo.
Ukuqapha kunconywa kwiziguli esezikhulile nabantu abane-pathologies yesibindi.
Ungayithatha kanjani i-Emoxipin Plus
Ukwethulwa kwekhambi ku / m kanye / ku kwenziwa nge-Drip. Ilungiselelwe ngokushesha ngaphambi kwenqubo emizuzwini engama-5-7. Umthamo ophakanyisiwe wokwelapha kufanele uchitheke ku-isotonic sodium chloride. Umthamo unqunywa ngawodwana. Imiyalo ikhombisa uhlobo lokulinganiselwa lwesilinganiso:
- phakathi naphakathi - 10 mg / kg yesisindo 1 isikhathi ngosuku;
- intramuscularly - akukho ngaphezu kwama-60 mg kanye izikhathi ezingama-2-3 ngosuku.
Isikhathi sokusetshenziswa siyizinsuku eziyi-10-30. Ukuthola imiphumela ephezulu, kunconyelwa ukuphatha isixazululo ngaphakathi kwezinsuku ezingama-5-8, sonke isikhathi, ukuphatha umuthi nge-intramuscularly.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-10.jpg)
I-Emoxipin yezidakamizwa iyatholakala kuma-ampoules.
Ukufakwa kwamaconsi kwenziwa ku-conjunctival sac. Ngaphambi kwenqubo, kuyadingeka ukuvula ibhodlela, gqoka i-dispenser futhi unikine ngamandla. Isitsha siphendulwe sabheka phansi. Ukucindezela i-dispenser kuzokwenza kube lula ukubala inani elidingekayo lamaconsi. Isimo sokwelapha isiguli esikhulile sihla kathathu ngosuku. Inkambo yokwelashwa ezimweni eziningi yizinsuku ezingama-30. Uma kunesidingo, inganwetshwa ize ifinyelele ezinsukwini ezingama-180.
Ngoshukela
Iziguli ezinesifo sikashukela zingadinga ukulungiswa komthamo. Ukwelashwa kufanele kuqalwe ngomthamo wesigamu.
Imiphumela emibi ye-Emoxipin Plus
Umuthi onokulawulwa okungafanele noma obedlula okujwayelekile ukwelashwa ucasisa ukuthuthukiswa kwemiphumela emibi evela ohlelweni lwezinzwa oluphakathi nezitho zangaphakathi. Lokhu kufaka phakathi:
- izinzwa zobuhlungu kanye nokuvutha kwemizwa endaweni yomjovo;
- ukozela
- ukweqile;
- isifo se-metabolic (akuvamile);
- ukwanda kwengcindezi yegazi;
- ukukhuphuka kwenhliziyo;
- i-migraine
- umuzwa ovuthayo emehlweni;
- ukulunywa
- hyperemia.
Ukungezwani komzimba kubonwa kuma-26% eziguli. Zibonakala njengokubomvu esikhunjeni, emaphashini nasekuwuncineni.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-11.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-12.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-13.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-14.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-15.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-16.jpg)
Imiyalo ekhethekile
Ukuphathwa kwe-Intravenous kudinga ukuqapha ngokucophelela umfutho wegazi nokuqunjelwa kwegazi. Ngokusebenzisa kanye kanyekanye amaconsi wamehlo kubakhiqizi abahlukahlukene, ukufakwa kwe-angioprotector kunconyelwe ukwenziwa ekugcineni. Isikhathi sokuphakathi kokufakwa kufanele sibe imizuzu engama-20-25.
Ngesikhathi sokuqhaqhazela, amafomu amagwebu, angathinti ikhwalithi yomuthi. Foam inyamalala ngokwayo ngemuva kwemizuzwana eyi-15-30. Ukusetshenziswa isikhathi eside kwesidakamizwa kuthinta izinga le-lycopene (antioxidant, i-carotenoid pigment) emzimbeni.
Sebenzisa ebudaleni
Ezigulini esezikhulile, kungcono ukusebenzisa umjovo we-intramuscular ukugwema ukwakheka kwe-hematomas. Kunconywe ukusetshenziswa kwengxenye yemithamo.
Ukunquma i-Emoxipin Plus ezinganeni
Imithi (kungakhathalekile ukuthi ifomu lomthamo) ayinqunyelwe iziguli ezingaphansi kweminyaka engu-18.
Sebenzisa ngesikhathi sokukhulelwa nokukhishwa komzimba
Ukusetshenziswa kwesidakamizwa ngesikhathi sokukhulelwa nokuzala ingane akuvunyelwe ngokuphelele.
Ukweqisa kwe-Emoxipin Plus
Amacala okweqa ngokweqile ayivelakancane. Zihambisana nezimpawu zobuntu, kufaka phakathi isicanucanu, ukuhlanza, izinhlungu esiswini. Ukwelashwa okubonakalayo, ukuphathwa kwama-enterosorbents kanye ne-gastric lavage kuyadingeka.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu-23.jpg)
Umuthi i-Emoxipin (kungakhathalekile ukuthi ifomu lomthamo) awunqunyelwe ezigulini ezingaphansi kweminyaka engu-18.
Ukuxhumana nezinye izidakamizwa
Izisombululo ze-infusion azikhuthazwanga ukuthi zisetshenziswe kanyekanye namanye amalungiselelo we-vascular, ama-antibiotics kanye ne-proton pump inhibitors. Izidakamizwa ezingenhla zinganciphisa umsebenzi kanye ne-bioavailability ye-angioprotector. Ukusetshenziswa kanyekanye kwezidakamizwa nezidakamizwa ezingama-antiviral kukhuthaza ukukhula kokuhluleka kwesibindi ngenxa yomthwalo omkhulu kulesi sitho.
Amaconsi wamehlo angahlanganiswa nemithi ye-herbal (i-ginkgo biloba ekhishwe, i-blueberries) ethuthukisa umbono. Ukusetshenziswa kwamaconsi kungahambisana nemijovo ye-intramuscular of amavithamini.
Ukuhambisana notshwala
Umuthi awuhambelani ne-ethanol. Ukusetshenziswa kotshwala ngesikhathi sokwelashwa kwenqatshelwe ngokuphelele.
Ama-Analog
I-angioprotector inezindawo eziningi ezinomphumela ofanayo wokwelapha. Abalingani abaningi abenziwe ngaphakathi basendleleni ephakathi yamanani futhi bayatholakala kwiziguli eziningi. Lokhu kufaka phakathi:
- I-Emoxipin-Akti. Analogue yesakhiwo yoqobo. Into efanayo esebenzayo ekuqoqweni okuncane inomphumela we-angioprotective ne-antioxidant emzimbeni wesiguli. Ukusetshenziswa ngezinjongo zokuvimbela nokwelapha kuvunyelwe ku-ophthalmology, inhliziyo and neurosurgery. Kukhona ukuphambana. Intengo emakhemisi isuka kuma-ruble angama-200.
- Isazi se-Emoxy. Kutholakala ngesimo samaconsi e-ophthalmic. Isetjenziswa ngaphezulu ngezinhloso zokwelapha kuphela ezigulini ezindala. Ukwakheka kuqukethe i-methylethylpyridinol hydrochloride (10 mg). Mhlawumbe ukuthuthukiswa kwemiphumela emibi. Izindleko - kusuka kuma-ruble angama-90.
- I-Cardioxypine. I-angioprotector enamandla esisiza ukunciphisa ukuncipha kwemithambo yegazi. Ngokusetshenziswa njalo, izitsha zobuchopho ziba namandla ngokwengeziwe kwi-hypoxia. Ukusetshenziswa ngezinjongo zokwelapha kanye ne-prophylactic kwenziwa ngemvume kadokotela. Intengo - kusuka kuma-ruble angama-250.
- Methylethylpyridinol-Eskom. Analogue yezakhiwo zesidakamizwa sokuqala. Ukuqanjwa kufana ngokuphelele, njengoba kunjalo izinkomba zokusetshenziswa. Imiphumela emibi nokuphikisana okuphelele kubekwe kwimiyalo. Izindleko emakhemisi zivela kuma-ruble ayi-143.
Ukukhethwa komuntu obambele esikhundleni kwenziwa ngudokotela oholayo uma isiguli sinokuphikisana ngokuphelele nokusetshenziswa komuthi ngenhloso yokuvimbela nokwelapha.
Imibandela yekhefu lekhemisi
Dinga umuthi weholide emakhemisi.
Ngingakwazi ukuthenga ngaphandle kadokotela
Umuthi awunakuthengwa ngaphandle kwencwadi kadokotela ekhethekile.
Intengo ye-Emoxipin Plus
Izindleko zomuthi emakhemisi zivela kuma-ruble ayi-135.
Izimo zokugcina zomuthi
Indawo yokubeka kufanele ibe yinhle futhi ibe mnyama, ingafinyeleleki ezinganeni nasezilwaneni.
Isikhathi sokuphelelwa yisikhathi
Impilo yeshalofu yesisombululo yizinyanga ezingama-36, amaconsi e-ophthalmic - azidluli izinyanga ezingama-24.
![](http://img.diabetesentity.com/img/sayd-2020/1442/preparat-emoksipin-plyus-instrukciya-po-primeneniyu.png)
I-Cardioxypine iyi-analogue ye-Emoxipin yokulungiselela.
Umkhiqizi
I-Enzyme (Russia), Tallinn Pharmaceutical Plant (Estonia).
Ukubuyekezwa kwe-Emoxipin Plus
U-Evgenia Bogorodova, udokotela wezifo zenhliziyo, iYekaterinburg
Lapho ngisebenza, ngisebenzisa lo muthi isikhathi esingaphezu kweminyaka emi-5. Nginikeza iziguli ezimweni ezimbi kakhulu, zinamandla. I-Angioprotector ithuthukisa i-microcirculation yegazi futhi inomphumela onenzuzo ebuchosheni. Ngokusebenzisa njalo, ubungozi bokuhlaselwa yisifo senhliziyo nemivimbo kuncishiswa kaningana. Ngaphezu kwalokho, umuthi uvikela ubuchopho ekubulaleni i-oksijini.
Imiphumela emibi yenzeka ezigulini eziningi ngenxa yezimpawu zomzimba ngamunye. Imvamisa kakhulu le yimiphumela yokungezwani komzimba (i-acne, redness yezingqimba ezingehla ze-dermis) ne-dyspepsia Isiguli siba nobuhlungu be-epigastric, isicanucanu, nokuhlanza. Ukwelashwa okubonakalayo kufanele kukhethwe ngokucophelela, awukwazi ukukhetha umuthi ngokwakho.
U-Elena, oneminyaka engama-46, eSt
Ngezokwelapha ngasebenzisa amaconsi e-ophthalmic. IGlaucoma yatholakala eminyakeni eminingana eyedlule, futhi yelashwa isikhathi eside. Imithambo yegazi ibe buthaka, waqala wabona ukuthi ama-capillaries ahlala eqhuma. Ama-hematomas kwabamhlophe bamehlo anyamalala isikhathi eside, amaconsi ajwayelekile awazange asize okuningi. Ngenxa yalokhu, umbono wawela, iso elilodwa laba nzima ukubona. Ngaphendukela ku-ophthalmologist ukuthola izeluleko, weluleka i-angioprotector eyenziwe ekhaya.
Ngathenga umuthi onikezwe umuthi. Kusetshenziswe ngokwemiyalo - kudonsa kabili kanye esweni ngalinye kabili ngosuku. Imiphumela emibi yavela ngosuku lokuqala. Amehlo akhe ayeshayekile futhi enamanzi. Kwavela amabala abomvu ezinqeni. Ngangesaba ukusebenzisa amafutha e-antihistamine, ngathambisa izinkophe ngo-ukhilimu wengane. Naphezu kokwenqatshwa, umuthi wasiza ngokushesha. I-hematoma ixazululwe ngokuphelele ezinsukwini ezi-2, umbono wabuyiselwa ngokuphelele ngemuva kwezinsuku ezingama-4.