Ungayisebenzisa kanjani isidakamizwa i-Aspirin 100?

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I-Aspirin (ASA), ngenxa yezindlela zayo zokwelapha, iyingxenye yemithi ethile enemiphumela ehlukahlukene. Izidakamizwa ezingezona ezombumbulu ezine-ASA zitholakala ngezindlela ezahlukahlukene, kufaka phakathi ama-suppositories wezingane ezisanda kuzalwa nezingane ezingaphansi kweminyaka engu-3.

Ukusetshenziswa kwemithi yalesi sigaba kwenziwa njengoba kushiwo udokotela, ikakhulukazi izingane kanye neziguli esezikhulile.

Ukusetshenziswa isikhathi eside kwe-ASA kungavusa ukuthuthukiswa kwemiphumela emibi eminingi ephazamisa ukusebenza okujwayelekile kwezitho zangaphakathi nohlelo lwezinzwa oluphakathi.

Igama Lezwe elingafanele

I-INN yesidakamizwa yi-acetylsalicylic acid.

I-Aspirin (ASA), ngenxa yezindlela zayo zokwelapha, iyingxenye yemithi ethile enemiphumela ehlukahlukene.

I-ATX

Umuthi wanikezwa ikhodi ye-ATX - N02BA01 nenombolo yokubhalisa - N013664 / 01-131207.

Khipha amafomu nokwakheka

Zonke izinhlobo zezindlela zemithamo, ezibandakanya i-ASA, ziyahlukahluka ekuqoqweni kwento esebenzayo nabazitholelayo. Okuqukethwe kwento esemqoka ngezindlela eziningi kungu-100 mg. Ezidakamizweni ezisetshenziselwa izinjongo zokwelapha izifo zezifo zenhliziyo, ukuhlangana kwento esebenzayo kufinyelela ku-50 mg.

Kusetshenziswa umuthi wezifo zesistimu yenhliziyo, ukuqoqwa kwento esebenzayo kufinyelela ku-50 mg.

Umuthi uyatholakala ngesimo:

  • amaphilisi
  • amaphilisi.

Izithako kanye nama-okhilimu ane-acetylsalicylic acid akhiqizwa ngamabhizinisi wezimonyo. Ukusetshenziswa kwezidakamizwa ezisetshenziselwa kwangaphandle kungenzeka ngezifo zesikhumba, kuhambisana nenqubo yokuvuvukala.

Amaphilisi

Amathebulethi e-biconvex amhlophe, ayindilinga anemiphetho edwetshwe kaningi i-facet futhi asengozini. Ngokuya ngomkhiqizi, amaphilisi angaba namalogo noma okuqoshiwe. Izinto ezisizayo ekwakhiweni kwefomu lomthamo:

  • isitashi sesitshalo (ummbila);
  • i-microcrystalline cellulose;
  • crospovidone.

Kuyathengiswa amaphilisi e-ufanisi.

Kuthengiswa amaphilisi we-Aspirin.

Zibekwe emaphaketheni amaselula noma amashubhu epulasitiki ngenani lama-10 ama-pcs. Inani lamabhulokhi epakethe lamakhadibhodi e-1 yi-2-10 ama-pcs. Imiyalo yokusebenzisa iyatholakala kwiphakeji ngayinye.

Amaconsi

I-ASA ngendlela yamaconsi ikhiqizwa ukukhathazeka kwemithi yaseJalimane. Kubukeka njengoketshezi olungacacile, olungenamibala onephunga elingathathi hlangothi nokunambitheka okumunyu. Isiraphu ithululelwa emabhodleleni engilazi afakwe i-dispenser.

Ngaphezu kwe-ASA, kumaconsi kukhona:

  • amanzi ahlanziwe;
  • ukukhipha peppermint;
  • ethanol.

Amabhodlela athengiswa emabhokisini amakhadibhodi.

Powder

Le ndlela yokukhishwa ayikho. Kukhona ama-analogues ngendlela ye-powder equkethe i-acetylsalicylic acid.

Kukhona ama-analogues ngendlela ye-powder equkethe i-acetylsalicylic acid.

Isixazululo

Le ndlela yokukhishwa ayikho.

Amakhandlela

Ifomu le-capsule alitholakali ukuthi lithengiswa.

Amafutha

Izithambisi zokwelapha, ukuqoqwa kwe-ASA okuyi-100 mg, akutholakali kuthengiswa.

Amakhandlela

I-Aspirin 100 ngendlela yamakhandlela ayitholakali. Ukulungiswa kwasekuqaleni kune-analogues ngendlela yama-suppositories.

Isenzo se-Pharmacological

Umuthi ungowesigaba sezidakamizwa ezingezona ezokwelapha ezibangela ukuvuvukala.

I-ejenti ye-antiplatelet, ngaphezu kokulwa nokuvuvukala, inomphumela we-antipyretic emzimbeni futhi inciphisa igazi.

Ngokusetshenziswa njalo, umuthi usebenza njenge-inhibitor yamapuleti, unciphisa ukuhlanganiswa kwawo futhi uvimbele ukwakheka kwe-thromboxane.

Ngokusetshenziswa njalo, into esebenzayo isebenza njenge-inhibitor yamaplatelet, inciphisa ukuhlanganiswa kwabo futhi ivimbele ukwakheka kwe-thromboxane.

Umuthi wemiphumela ehlukahlukene onomphumela omude wokwelapha. Ukwakheka kwe-cycloo oxygenase kuyaphazamiseka.

I-Pharmacokinetics

Inqubo yokubola ishesha. Uma ifomu lomthamo (amaphilisi we-enteric noma we-effeedcent) lingena, ukumunca kwenzeka ngemuva kwemizuzu engama-20. I-acetylsalicylic acid iguqulwa kancane kancane ibe acid acid. Ukuhlungwa okuphezulu kwe-ASA esegazini lesiguli ngemuva kokutholakala komthamo wokuqala emva kwemizuzu engama-20-25. Ulwelwesi lwe-enteric lubambezela ukuqhekeka kwethebhulethi, okwenzeka ezingxenyeni ezingenhla zamathumbu amancane.

Umuthi ulolongwa esibindini. Ama-Metabolites enziwe ngale nqubo ancishwa umsebenzi. I-Excretion yenziwa izinso, iningi lazo likhishwa emchameni. Akukho ngaphezu kwe-2% yezidakamizwa ezishiya umzimba ungashintshiwe. Into esemqoka ibopha amaprotheni egazi ngama-62-65%.

Okusizayo

Ukusetshenziswa komuthi kwenziwa ngenhloso yokuvimbela nokwelapha. Izinkomba eziphambili zokusebenzisa yilezi:

  • ukuphazamiseka kokujikeleza kwegazi, kubandakanya nesifo sohlangothi;
  • infarction myocardial;
  • i-thromboembolism;
  • venous thrombosis;
  • izifo zesistimu yenhliziyo;
  • i-arthrosis;
  • ukutheleleka ngegciwane.
Izinkomba eziphambili zokusetshenziswa yiziphazamiso zokujikeleza kwegazi, kufaka phakathi unhlangothi.
Izinkomba eziphambili zokusetshenziswa yi-infyoction ye-myocardial.
Izinkomba eziphambili zokusetshenziswa yi-thromboembolism.
Izinkomba eziphambili zokusetshenziswa yizifo zohlelo lwethambo nenhliziyo.
Izinkomba eziphambili zokusetshenziswa yi-venous thrombosis.
Izinkomba eziphambili zokusetshenziswa yi-arthrosis.
Izinkomba eziphambili zokusetshenziswa yizifo ezibangelwa amagciwane.

Ukuvimbela nomuthi kungenzeka lapho iziguli zikhomba izici zobungozi, ezibandakanya:

  • isifo sikashukela mellitus;
  • ukukhuluphala kwamazinga ahlukahlukene;
  • izifo zamaphaphu ezibangelwa ukuhlukunyezwa kukagwayi;
  • hyperlipidemia;
  • ubudala.

Ukwelashwa kwezifo kusuka ohlwini ezinganeni ezine-acetylsalicylic acid kuvunyelwe ngezizathu zezempilo.

Contraindication

Ukuzwela kwesiguli entweni eyinhloko ekwakhekeni komuthi kubhekwa njengokuphambana okubalulekile. Futhi, umuthi unokwephulwa okuhlobene okuhlobene ngokuphelele.

Cabanga ngokuphelele:

  • isifuba somoya
  • diathesis;
  • ukwehluleka kwenhliziyo okukhulu;
  • umsebenzi wezinso ongonakalisiwe;
  • i-pathology yesibindi.

Ukuba khona kwe-contraindication ngokuphelele kwenza kungenzeki ukuthatha umuthi.

Ukuphikisana ngokuphelele nokuthatha i-Aspirin yisifo somoya.
Ukuphambana okuphelele kokuthathwa kwe-Aspirin kungukuguquguquka.
Ukwephula umthetho okuphelele kokuthatha i-Aspirin kubhekwa njengokwehluleka kwenhliziyo okukhulu.
Ukwephulwa okuphelele kokuthatha i-Aspirin kubhekwa njengokwehluleka kwezinso.
I-contraindication ngokuphelele yokuthatha umuthi yi-pathologies yesibindi.

Ngokunakekela

Ukuqapha kuyadingeka ezigulini ezine-contraindication ezihlobene. Lokhu kufaka ukukhulelwa, isikhathi sokuncelisa ibele, ubuntwana kanye nezifo zomgudu wesisu, kubandakanya nomlando wokuphuma kwegazi kwamathumbu.

Ukuhlaselwa isithuthwane kungabhekwa njengokwephula umthetho okulinganiselwe: ukubonwa ngudokotela ohambelayo kanye nokulungiswa kwendlela yemithamo kungadingeka.

Ungayithatha kanjani i-Aspirin 100

Ezigulini zabantu abadala, uhlobo lomthamo lunqunywa ngokuhlukile, kususelwa esimweni esivamile sesiguli. Zonke izinhlobo zemithamo zenzelwe ukuphathwa ngomlomo. Amaconsi kufanele ancibilikiswe inani elincane lewuketshezi, amaphilisi kufanele aphuculwe, agezwe phansi ngo-150 ml wamanzi.

Okungakanani

Imithamo yansuku zonke ayidluli kuma-300 mg. Ukuze kube lula, ochwepheshe batusa ukuthatha ithebhulethi engu-1 kathathu ngosuku.

Isikhathi esingakanani

Inkambo yokusebenzisa akufanele idlule izinsuku eziyi-10.

Ukuthatha umuthi wesifo sikashukela

Isifo sikashukela sidinga imithamo. Ukusetshenziswa kokuvimbela umuthi wesifo sikashukela kwenziwa ngaphansi kokuqondisa kukachwepheshe. Izinga lansuku zonke akufanele lidlule i-150 mg le-ASA.

Isifo sikashukela sidinga imithamo eyi-Aspirin.

Imiphumela emibi ye-Aspirin 100

Imiphumela emibi ikhula ngokusetshenziswa kabi komuthi noma ukungahambisani nemiyalelo yezokwelashwa. Babonwa engxenyeni yezitho zangaphakathi nohlelo lwezinzwa.

Amapheshana wesisu

Ukusuka emgudwini wokugaya ukudla, isiguli singakhula i-pancreatitis, i-gastritis, ukwakheka kwegesi ngokweqile emathunjini kanye nobuhlungu esifundeni se-epigastric. Ubungozi bokukhula kwesibindi sangaphakathi luyakhula.

Izitho zeHematopoietic

Kusukela ohlangothini lwe-anemia system ye-anemia, i-leukopenia, i-arrhythmias yenhliziyo, i-thrombocytopenia kanye ne-agranulocytosis kuyabonakala.

Isistimu yezinzwa ephakathi

Imiphumela emibi evela ohlelweni lwezinzwa oluphakathi ibonakaliswa ngesimo sokuzela, isiyezi, i-migraine ne-Huntington's syndrome.

Kusuka ohlelweni lomchamo

Imiphumela emibi ehambisana nohlelo lomchamo ivela ngenxa yokulimala kokuchama komchamo. Isiguli sihlakulela i-oliguria.

Imiphumela emibi evela ekuthatheni ingavela ngendlela yobuhlungu emgodini wokugaya ukudla, ubuhlungu esifundeni se-epigastric.
Imiphumela emibi evela ekwemukelweni ingenza i-anemia system ye-anemia, ukuphazamiseka kwesigqi senhliziyo.
Imiphumela emibi evela ohlelweni lwezinzwa oluphakathi ibonakaliswa ngendlela yesiyezi.
Imiphumela emibi ehambisana nohlelo lomchamo ivela ngenxa yokulimala kokuchama komchamo.

Allergies

Ukuvela kwe-allergic kubonakala njengokuqhuma esikhunjeni. Ukuqhekeka nokoma kwe-mucosa yamakhala nezimpawu zomlomo kungabhekwa ngemiphumela emibi.

Umthelela ekhonweni lokulawula izindlela

Ukusetshenziswa isikhathi eside kwe-acetylsalicylic acid kungadala ukozela nokwehla kwezimpendulo ze-psychomotor. Kunconywa ukwenqaba ukushayela izimoto nezinye izindlela zesikhathi sokwelashwa nomuthi.

Imiyalo ekhethekile

Ukusetshenziswa komuthi kufanele kwenziwe ngokuqinile ngokwemiyalo. Amatafula kufanele agezwe kuphela ngamanzi - iziphuzo ezinekhabhoni, ikhofi netiye azilungele lezi zinhloso. Ukwelashwa ngomuthi akudingi ukubuyekezwa kokudla nokudla.

Ukunquma u-Aspirin ezinganeni eziyi-100

Iminyaka yezingane kungukuphula umthetho okuhlobene; uhlelo lokusebenza luvunyelwe kusuka eminyakeni engu-6.

I-Aspirin neParacetamol - UDkt Komarovsky
Ukuphila okuhle! Umlingo Aspirin. (09/23/2016)

Sebenzisa ngesikhathi sokukhulelwa nokukhishwa komzimba

Imithi ingathinta ukukhula kwengane. Ukusetshenziswa kwomuthi ngesikhathi sokuncelisa ibele nokukhulelwa kwenziwa ngokwezinkomba ezibalulekile.

Sebenzisa ebudaleni

Iziguli asebekhulile bayelulekwa ukuthi baphuze lo muthi ngemithamo yemigqa.

Ukweqiwa kwe-Aspirin 100

Izimpawu ezisetshenziswayo zokweqisa ngokweqile zivezwa njenge-dyspepsia, ikhanda, i-hypokalemia, ukuhlanza kanye nokukhubazeka okubukwayo.

Usizo lokuqala luqukethe ukuhanjiswa kwesisu nokuphathwa ngomlomo kwama-enterosorbents. Uma isimo sesiguli singazange sithuthuke, kuyadingeka ukuxhumana nesikhungo sezokwelapha.

Ukuxhumana nezinye izidakamizwa

Ukusetshenziswa kanyekanye kwe-acetylsalicylic acid nezinye izidakamizwa akwamukeleki. Ukuhlaziywa kanye ne-ASA kwandisa ingozi yokopha kwesisu.

Ukuhlaziywa kanye ne-ASA kwandisa ingozi yokopha kwesisu.

Ama-Thrombolytics, amanye ama-antiplatelet agents, ama-diuretics, ama-salicylate derivatives, ama-digoxin awahambisani nomuthi.

I-Ibuprofen yehlisa umsebenzi we-ASA.

Ukusetshenziswa okuyinkimbinkimbi kwezidakamizwa ze-hypoglycemic kanye ne-ASA kufanele kwenziwe ngaphansi kokuqashwa kukadokotela oholayo.

Ukuhambisana notshwala

Ukusetshenziswa kotshwala ngasikhathi sinye nomuthi akufakiwe. I-Ethanol kanye ne-ASA ibangela ukudakwa okukhulu.

Ama-Analog

Umuthi unezinto zokufaka eziningana ezinokuphilisa okufana nokwangempela.

Analogs ifaka:

  1. Brilinta. Umuthi ukhiqizwa eSweden, uyatholakala ngesimo samathebulethi. Isisekelo somuthi yi-ticagrelor mannitol. I-ejenti ye-antiplatelet ine-contraindication, eyinhloko okuyizikhathi zokuzala kwengane nokungabekezelelani ngakunye. Izindleko zomuthi zivela kuma-ruble angama-4,000.
  2. I-Plavix. Umuthi waseFrance. Ithebhulethi eyi-1 iqukethe kufika ku-300 mg wento esebenzayo - i-clopidogrel. Imemezele izakhiwo ze-antiplatelet, ilawula ukuhlanganiswa kweplatelet. Intengo emakhemisi iqala kuma-ruble ayi-1,500.
  3. I-Thrombo Ass. Umuthi wase-Austrian, i-analogue esondelene kakhulu yoqobo. Ukuhlushwa kwe-acetylsalicylic acid kumathebulethi eStrombo Ass kungama-50 mg. Izindleko zezidakamizwa ezingezona ze-steroidal zokulwa nokuvuvukala emakhemisi ezivela kuma-ruble angama-70.
Izinkomba ze-Aspirin
I-Plavix "Yangempela noma mbumbulu?"

Analogs akhethiwe uma isiguli has contraindication ukusetshenziswa kwangempela.

Imibandela yekhefu lekhemisi

I-ASA (kufaka phakathi ifomu le-Cardio) ayidingi ukunikezwa umuthi kusuka kumakhemisi.

Ngingakwazi ukuthenga ngaphandle kadokotela

Imithi ingathengwa ngaphandle kwemithi kadokotela.

Intengo ye-Aspirin 100

Umuthi osokhemisi ubiza ama-ruble ayi-100-180.

Izimo zokugcina zomuthi

Indawo yokugcina noma yiliphi ifomu lomthamo kufanele yomile, ipholile futhi iphephe ezilwaneni nasezinganeni.

Isikhathi sokuphelelwa yisikhathi

Ukupakisha ngomuthi kufanele kugcinwe iminyaka engu-5 kusukela ngosuku lokwenziwa kwawo.

Umkhiqizi

EGermany, iBayer Beiterfeld GmbH. Le nhlangano inamagatsha eSwitzerland.

I-Brilinta iyi-analog ye-Aspirin. Izindleko zomuthi zivela kuma-ruble angama-4,000.
I-Plavix iyi-analogue ye-Aspirin. Intengo emakhemisi iqala kusuka kuma-ruble ayi-1,500.
I-Thrombo Ass iyi-analog ye-Aspirin. Izindleko zezidakamizwa kumakhemisi kusuka kuma-ruble angama-70.

Ukubuyekezwa ku-Aspirin 100

I-Kasatkina Angelina, isazi sezinhliziyo, uKrasnodar

Ngincoma umuthi ezigulini iminyaka engu-7. Izici zemithi ukuthi zingasetshenziselwa izinjongo zokwelapha kanye ne-prophylactic. Imvamisa ngisebenzisa umuthi ezingozini ze-cerebrovascular, ekuvinjelweni kokuhlaselwa yisifo senhliziyo nemivimbo. Ama-pluses amakhulu ayakwazi ukubekezelela umuthi ezigulini ngentengo ephansi.

Imiphumela emibi ezigulini eziningi ivela njengokuphendula komzimba. Kungenzeka unciphise ingozi yokwenqatshwa yi-ASK isiguli uma isiguli sigcina ngokucophelela yonke imiyalo kadokotela. Uhlobo lwedosi ekhethwe kahle icishe ikuqede ngokuphelele ukuthuthukiswa kwemiphumela emibi.

UGrigory, oneminyaka engama-57 ubudala, eSt

Umuthi owabekwa eminyakeni eyi-4 eyedlule. Wahlaselwa unhlangothi, isimo sakhe besingesihle, kwakukhona ubuthakathaka, ikhanda elibi. Ucwaningo luveze ukuthi kunezingozi zokushaywa kwegazi. Babeka i-stent, kufanele ibe nesiphambano esihle. I-Sensitivity ivele ezidakamizweni zezifo zohlelo lwethambo nenhliziyo, isidingo esiphuthumayo sokuxazulula inkinga.

I-cardiopreparation isebenze kahle, ayengalindele nakancane umphumela onjalo. Isimo saba ngcono, ama-migraines anyamalala. Ukuhlaziywa kuhle kakhulu. Izinsuku zokuqala ezimbalwa zaqaphela imiphumela emibi. Ukuqhakaza kwavela engxenyeni yesisu namathumbu; ukuqunjelwa kwaphazamiseka ezinsukwini ezimbili zokuqala. Angiphathanga lutho ngasikhathi sinye, ukugula kuhambile ngedwa.

U-Evelina, oneminyaka engama-24 ubudala, e-Ekaterinburg

Ubaba eminyakeni engu-2 edlule wahlaselwa unhlangothi. Ngenxa yobudala, imiphumela yayinkulu: ukuzwela kwengalo yangakwesobunxele kunyamalale futhi ukukhuluma kukhubazeke kancane. Inqubo yokuvuselela kabusha yathatha isikhathi esingaphezu kwenyanga. Kepha ubaba ucishe walulama ngokuphelele.Bypassed inani elikhulu lochwepheshe abeluleke ukuthi bakhethe ithuluzi eliphumelela kakhulu elivimbela ukwakheka kwezigaba zegazi. Umuthi kufanele unciphise igazi futhi ulenze lingabonakali kancane. Ngemuva kokusesha isikhathi eside, sahlala kwi-ejenti ye-antiplatelet, efaka i-ASA.

Udinga ukuyiphuza nsuku zonke, ngaphandle kokuphazamisa ukungena kokudla: Ithebhulethi le-1 kathathu ngosuku. Kuhle ukuphuza umuthi ngasikhathi sinye. Izinsuku zokuqala ezi-3, ochwepheshe babone ukusabela komzimba, udokotela wesifunda wayevakashela njalo. Imiphumela emibi ibe yesikhashana. Izinduna zavela esikhunjeni kanye nokuyalunywa kwayo. I-antihistamine yamafutha yasiza ukuqeda ukungaphenduki komzimba.

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