I-Pentoxifylline 100 yesifo sikashukela

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Ithuluzi libuyisela ukuhamba kwegazi okujwayelekile ngama-microvessels. Ivimbela ukunamathela kwe-platelet, ithuthukisa ukuhamba kwegazi. Isetshenziselwa ukuphazamiseka kokujikeleza kwegazi.

Igama Lezwe elingafanele

I-Pentoxifylline

I-Pentoxifylline 100 ibuyisela ukuhamba kwegazi okujwayelekile ngokusebenzisa ama-microvessels.

I-ATX

I-ะก04AD03

Khipha amafomu nokwakheka

Umenzi ukhiqiza umuthi ngendlela yamathebulethi e-enteric. Umuthi osebenzayo yi-pentoxifylline ngenani le-100 mg.

Amaphilisi

Kuhlanganiswe izingcezu ezingama-20. emaphaketheni.

Izindlela ezingekho

Uhlobo olungatholakali lokukhululwa - amaconsi namaphilisi.

Isenzo se-Pharmacological

I-Pentoxifylline ivimbela isenzo se-phosphodiesterase, yehlisa inani le-calcium ngaphakathi kwamangqamuzana, futhi ivimbele ukuhlanganiswa kweplatelet. Umuthi uvuselela imithambo yegazi, kusiza ukuhamba kwegazi ngokusebenzisa ama-microvessels, futhi kunomthelela ekugcwalisweni kwezitho ezine-oxygen.

I-Pentoxifylline 100 igxilisa imithambo yegazi, isiza ukuhamba kwegazi ngokusebenzisa ama-microvessels.

I-Pharmacokinetics

Kusuka emgudwini wokugaya udonswa ngokushesha. Ngenqubo yokugayeka kokudla emzimbeni, kwakheka izakhi ezisebenzayo esibindini. Ngemuva kwemizuzu engama-60, ukuqoqwa kwezithako ezisebenzayo egazini kufinyelela inani lazo eliphezulu. Isigamu sikhishwe emzimbeni ngemuva kwamahora we-1-2. Kukhiqizwa umchamo nezindunduma.

Yini esiza?

Ithuluzi lichaziwe ezimweni ezinjalo:

  • ukuphazamiseka kokujikeleza kwegazi lapho kukhona ukulimala kwamangqamuzana obuchopho, isifo sokuqina kwemizwa, noma isifo sikashukela;
  • ukonakala kwe-microcirculation ngokumelene ne-spasm of artery and arterioles (isifo sikaRaynaud);
  • ingozi ye-cerebrovascular eyingozi;
  • isifo se-artery se-artery;
  • i-necrosis yezicubu zomzimba;
  • ukulimala kwemithambo yemilenze;
  • izilonda ze-trophic;
  • ukwehluleka kokujikeleza kwe-choroid yeso;
  • ukonakala komsebenzi wokuzwa kwezimpawu ngenxa yokuphazamiseka kwemithambo yegazi.
IPentoxifylline 100 imiselwe isifo sikaRaynaud.
I-Pentoxifylline 100 ibekelwe ingozi yengozi yokuqina kwesibindi.
IPentoxifylline 100 imiselwe umonakalo emithanjeni yemilenze.

Umuthi usetshenziselwa ukuthuthukisa ukondleka kwezicubu futhi ubuyisele i-microcirculation nge-vein thrombosis ejulile, i-frostbite.

Contraindication

Umuthi uphambaniswe neziguli ngama-pathologies alandelayo:

  • ukungabekezeleli lesi sidakamizwa, kanye ne-hypersensitivity ku-caffeine, theophylline, theobromine;
  • i-corrhea hemorrhage;
  • isikhathi sokukhulelwa nokukhulelwa;
  • ukopha kakhulu;
  • ukopha kwemithambo ye-retinal;
  • izingane nentsha engaphansi kweminyaka engu-18.

Ithebhulethi alinqunyelwe ukwephula okunamandla kokuhlinzekelwa kwegazi emisipha yenhliziyo.

Ngokunakekela

Kunqunywa ngokuqapha ezigulini ezinokwehluleka okungapheli kwenhliziyo, ukusebenza kwe-renal kabi kanye ne-hepatic, umfutho wegazi ophansi, isilonda se-peptic sesisu kanye ne-duodenum. Iziguli ezisanda kwenziwa ukuhlinzwa kufanele zisetshenziswe ngaphansi kokuhlolwa udokotela.

Ngokuqapha, iPentoxifylline 100 ibekelwe iziguli ezinokwehluleka kwenhliziyo okuhlala njalo.

Ungayithatha kanjani i-pentoxifylline 100?

Amathebulethi athathwa ngemuva kokudla. Umthamo wokuqala amaphilisi ama-2 kathathu ngosuku. Unganciphisa umthamo ngemuva kwezinsuku ezingama-7-14 ukuya ku-100 mg. Ukwehluleka okungapheli kwezinso, udinga ukuthatha umuthi engxenyeni yesigamu. Umthamo wansuku zonke akufanele ube ngaphezu kwe-1200 mg. Isikhathi sokwelashwa sisuka ezinyangeni ezi-1 kuye kwezingu-3.

Ngoshukela

I-Pentoxifylline ingabhekelwa isifo sikashukela, ngoba ibhekana ngempumelelo nezinkinga eziningi zalesi sifo. Umthamo ukhethiwe ngokuhlukile ngokuya kobunzima besifo kanye nomphumela wokwamukelwa.

Umthamo wokwakha umzimba

Lesi sidakamizwa kwesinye isikhathi sisetshenziswa ngaphambi kokuqeqeshwa ngoba sisiza izicubu ukuba zigcwale kahle ngegazi futhi ziqhamuke kakhulu. Umuthi uthathwa uhhafu wehora ngaphambi kokuqeqeshwa. Umthamo onconyiwe amaphilisi ama-2 kabili ngosuku. Umthamo omkhulu yi-1200 mg. Ungasithatha isidakamizwa isikhathi esingaphezu kwenyanga, bese udinga ukuthatha ikhefu.

Imiphumela emibi yePentoxifylline 100

Ithuluzi libekezelelwa kahle ngumzimba, kepha futhi linemiphumela emibi.

I-Pentoxifylline ingabhekelwa isifo sikashukela.

Amapheshana wesisu

Ukwehla kwesifiso sokudla, ukuphazamiseka okuhlukahlukene kokuwohloka, ukuvuvukala kogange lwe-gallbladder, umsebenzi owandisiwe wama-enzyme wesibindi, ulwelwesi lwe-mucous lomlomo olomile.

Izitho zeHematopoietic

Yehla ngenani lama-leukocytes, izinkomba ezincishisiwe zazo zonke izinhlobo zamangqamuzana egazi, ukuncipha kokuqukethwe kwe-fibrinogen. Kusukela ohlangothini lwe-CCC, kukhona ukwehla komfutho wegazi, ukuthuthukiswa kwe-angina pectoris, i-Cardialgia, i-tachycardia.

Isistimu yezinzwa ephakathi

Ubuhlungu bekhanda buphawuliwe. Kwesinye isikhathi kuba nomuzwa wokukhathazeka, isiyezi, nokulala nokubuka ukonakala. Akuvamile, ukuvuvukala kolwelwesi lobuchopho nentambo yomgogodla.

Allergies

Ukulunywa, okhalweni, ukuvuvukala kwezicubu ezingaphansi kanye nezendlalelo ezijulile zesikhumba, nokuphawulwa kobuso obuso kuyaphawulwa. Ezimweni ezingavamile, ukuthatha lo muthi kuholela ku-anaphylaxis.

Umthelela ekhonweni lokulawula izindlela

Umuthi ungadala isiyezi, ukhubazeka okubukwayo, ukuqaqamba kwenhliziyo. Kufanele ishiywe isikhathi sokwelashwa kusuka ezimotweni zokushayela nezinqubo eziyinkimbinkimbi noma uqaphele.

Ngesikhathi sokulashwa, kubalulekile ukubheka umfutho wegazi.

Imiyalo ekhethekile

Ngemuva kokuhlinzwa, kuyadingeka ukulawula ukuqoqwa kwe-hemoglobin. Ngesikhathi sokulashwa, kubalulekile ukubheka umfutho wegazi. Uma abanesifo sikashukela bedinga ukuthatha izidakamizwa ukwehlisa amazinga kashukela, umthamo walesi sidakamizwa kufanele ulungiswe.

Ngokusetshenziswa kanyekanye kwezidakamizwa ezivimbela ukwakheka kwezigaba zegazi, kubalulekile ukubheka ukuvela kwegazi. Ukubhema kunciphisa ukusebenza kwalesi sidakamizwa.

Umthamo ekugugeni

Ebudaleni, umthamo kumele wehliswe, ngoba umuthi uthululwa kancane futhi kukhona ukwanda kwe-bioavailability.

Kungani iPentoxifylline ibekelwe izingane eziyi-100?

Lesi sidakamizwa asinqunyelwe izingane, ngoba imiphumela yaso emzimbeni wengane ayifundwanga.

Ngesikhathi sokukhulelwa nokuqunjelwa

Kuyavunyelwa ukusebenzisa umuthi kulezi zikhathi. Uma kunesidingo, ukuncelisa ibele kuyaphazamiseka.

I-overdose yePentoxifylline 100

Uma kwenzeka usebenzisa i-overdose, kuzovela lezi zimpawu ezilandelayo:

  • ubuqili;
  • isiyezi;
  • isimo sokulala;
  • ukungavikeleki kwemisipha etholakalayo;
  • ukukhohlisa
Nge-overdose, isiyezi.
Nge-overdose, kuvela isimo sokulala.
Uma kwenzeka kuba ne-overdose, ukutholakala kwemisipha ngokuzithandela kuyabonakala.

Lapho kuvela izimpawu zokuqala, udinga ukuhlanza isisu, uthathe namalahle ocushiwe. Uma ukuvela kuhlangana, udokotela angayala ama-anticonvulsants.

Ukuxhumana nezinye izidakamizwa

Ukuqiniswa komphumela kwenzeka ngokusetshenziswa kanyekanye kwezidakamizwa ezithinta ukuqina kwegazi. Izidakamizwa zokucindezela, ukunciphisa ukugcwala kwe-glucose, i-valproic acid kanye nemithi elwa namagciwane aqala ukuthatha isinyathelo ngokushesha ngaphansi kwesenzo se-pentoxifylline.

Ukusetshenziswa kwalesi sidakamizwa namanye ama-xanthines kuholela ekubukekeni kokugula kwengqondo.

I-Cimetidine inyusa inani le-pentoxifylline egazini futhi lokhu kungaholela ekuphendukeni okubi. I-Theophylline kufanele ithathwe ngokuqapha.

Ukuhambisana notshwala

Ukuphuza utshwala ngesikhathi sokwelashwa kwenqatshelwe. Ngaphandle kwalokho, ukusabela okungekuhle kuyaqina futhi ubuthi bomzimba nge-ethanol. Ukwelapha kungenzeka kungasebenzi.

Ama-Analog

Izidakamizwa ezilandelayo zingathengwa ekhemisi:

  • I-Flowerpot;
  • Pentilin;
  • I-Pentoxypharm;
  • Trenpental;
  • I-Flexital.
Izikhundla zePentoxifylline zingathengwa ekhemisi, kufaka neVasonite.
Izikhundla zePentoxifylline zingathengwa ekhemisi, kufaka phakathi iPentilin.
Izikhundla zePentoxifylline zitholakala ekhemisi, kufaka phakathi iFlexital.

Izidakamizwa ezifanayo ekwakheni umzimba yiTrental ne-Agapurin. Ngaphambi kokusebenzisa le mishanguzo, kungcono ukuvakashela udokotela.

Imibandela yekhefu lekhemisi

Kukhishwe ngomuthi

Ngingakwazi ukuthenga ngaphandle kadokotela?

Akunakwenzeka ukuthenga isidakamizwa ngaphandle kwemiyalelo kadokotela.

Intengo yePentoxifylline 100

Izindleko zokufaka umuthi zivela kuma-ruble angama-295.

Izimo zokugcina zomuthi

Ukuhlanganiswa ngamathebhulethi kufanele kunqunywe endaweni emnyama enamazinga okushisa afinyelela ku + 25 ° C.

Isikhathi sokuphelelwa yisikhathi

Impilo yeshelf iyiminyaka emithathu.

Umkhiqizi

I-Organika JSC, eRussia.

I-Pentoxifylline
Imiyalo yePentoxifylline

Ukubuyekezwa kwePentoxifylline 100

Odokotela neziguli bashiya ukubuyekezwa okuhle ngePentoxifylline 100. Babona umphumela osheshayo, intengo engabizi kanye nokusebenza kahle. Uma ulandela umthamo futhi uthatha ngokwemiyalo, imiphumela emibi ayibhekwa.

Odokotela

U-Ilya Korneev, i-phlebologist, Kemerovo.

Umuthi uthuthukisa isimo sohlelo lokuthinta kwenhliziyo. Isetshenziselwa ukwephula i-arcial or venous microcirculation. Kuhle ekwelapheni iziguli ezinezikhathi ezithile phakathi kokungabikho kokujikeleza kwegazi emikhawulweni ephansi. Ngesikhathi sokwelashwa, udinga ukukala ingcindezi njalo. Ngaphansi kwengcindezi encishisiwe, i-incl. ebudaleni, kubalulekile ukuqala ukuthatha ngomthamo oncishisiwe.

U-Angelina Tikhoplav, udokotela wezinhliziyo, uReutov.

Ithuluzi likhuthaza i-oxygenation yegazi. Ngemuva kokuphuza umuthi, imithambo iphumule, i-myocardium iqala ukuthola umoya-mpilo omningi, imithambo yenhliziyo iyanda, ithoni yemisipha yokuphamba kanye naphakathi nendawo iyanda, ukuqina kwegobolondo langaphandle lamangqamuzana abomvu egazi kuyathuthuka. Ngincoma ukuthi ngiyeke ukubhema ngesikhathi sokuvuma, njengoba umkhuba omubi wehlisa umphumela wesithako esisebenzayo. Kunefomu elihlaselayo eliqukethe isisombululo se-sodium chloride ne-pentoxifylline.

Iziguli

U-Irina, oneminyaka engama-45, uTyumen.

Nikeza ithuluzi ekwelapheni okuyinkimbinkimbi kwe-vegetovascular dystonia. Usizo lwenzeka ezinsukwini ezimbalwa ngemuva kokuphathwa. Thatha cishe izinsuku eziyi-10. Ukuhlaselwa akwenzeki kaningi. Ithuluzi linciphisa ubuthakathaka, ikhanda kanye nesiyezi.

UKaterina, oneminyaka engama-33, eSt.

Kumamezala ngemuva kokudla umuthi, iziphetho zaqala ukuvuvukala kancane, futhi imithambo ye-varicose ayikhathazeki kangako. Ithuluzi linomphumela omuhle enhliziyweni nemithambo yegazi, ngakho-ke ukucindezela manje sekujwayelekile. Bathengile isidakamizwa i-Trental, kodwa base bethola nge-analogue eshibhile yaseRussia yePentoxifylline.

U-Andrey, oneminyaka engama-51, uSaratov.

Udokotela otolaryngologist unquma ithebhulethi eyi-1 kathathu ngosuku. Ngakhipha umsindo ekhanda lami, amehlo ami abe ngcono. Ngemuva kokwelashwa, udokotela wabika ukuthi isimo se-autonomic neva system sathuthuka. Ekupheleni kokwelashwa, waqala ukuphuza amaphilisi kabili ngosuku ngenxa yezinkinga zokucindezela. Wanelisekile ngomphumela.

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