Umuthi osuselwa ku-Pentoxifylline usiza ngokwezifiso i-microcirculation, unciphise ukuqina kwegazi futhi uthuthukise ukuhanjiswa kwezicubu ezinomsoco kanye nomoya-mpilo. I-Pentoxifylline neTrental ifaka leyo mithi. Banciphisa ngempumelelo ama-cramps, izinhlungu nokukhalinyelwa kwezikhathi ezithile, bandisa ibanga lokuhamba. Izidakamizwa ezinjalo zibhekwa njenge-analogues, futhi zingamalungu eqembu elilodwa lezemithi.
Isici sePentoxifylline
IPentoxifylline iyi-vasodilator yangaphandle. Isakhi saso esikhulu yi-pentoxifylline. Lesi sidakamizwa esisebenzayo esithuthukisa izakhiwo zegazi futhi sisiza nge-pathologies yemithambo yegazi. Inezindawo ezi-capillary-ezivikelayo nezivimbelayo, zandisa ukumelana kwe-capillary.
Umuthi uthinta imithambo ye-capillary, venous and arterial yomzimba womuntu. Ukusetshenziswa kwaso kusiza ukuthuthukisa ithoni yezicubu zokuphefumula futhi kuvimbele ukwakheka kwezigaxa zegazi. I-Pentoxifylline ithuthukisa ukuhamba kwegazi emithanjeni futhi ivikele izindonga zazo ngokunciphisa ukubukeka kwegazi futhi ikhuphule ukuqina kwamangqamuzana abomvu egazi.
Ngenkathi uthatha umuthi, isimo sezicubu nezitho zangaphakathi siyathuthuka ngenxa yokwanda komoya-mpilo kubo, izinqubo ze-bioelectric ebuchosheni ziyajwayelekile, nokujikeleza kwegazi ezindaweni eziphazamisekile kuyabuyiselwa.
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I-Pentoxifylline ithuthukisa izakhiwo zegazi futhi isiza ne-pathologies yemithambo yegazi.
Izinkomba zokusebenzisa i-pentoxifylline zingokulandelayo:
- i-arterial hypertension;
- ischemic stroke;
- ukungasebenzi kahle kwe-cerebrovascular;
- cholecystitis;
- imisipha ebushelelezi;
- dystrophy yemisipha;
- izilonda ze-trophic;
- urolithiasis;
- algodismenorea;
- ukwephulwa kokujikeleza kwegazi okujwayelekile emithanjeni yamehlo;
- i-encirchalatory encephalopathy;
- izifo zangaphakathi nezangaphakathi zezindlebe;
- isifuba somoya;
- isifo samathambo;
- Isifo sikaCrohn;
- i-psoriasis
- i-atherosclerotic encephalopathy.
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I-Pentoxifylline ayinakusetshenziswa ngokubekezelela umuntu ngamunye ezingxenyeni zomuthi. Ngaphezu kwalokho, kukhona okulandelayo okubhekiswa kokunye okusetshenziswayo:
- arrhythmia;
- umfutho wegazi ophansi;
- ukushaya kwe-hemorrhagic;
- isifo sokuqina kwemithambo yegazi emithanjeni yobuchopho;
- i-infarction ye-myocardial eyingozi kakhulu;
- i-retinal hemorrhage;
- ukukhulelwa nokuqunjelwa;
- izingane ezingaphansi kweminyaka engu-18.
Ukuthatha lo muthi kungaholela engcupheni yokopha, ngakho-ke akunconywa ukuthi uyise ezigulini ngemuva kokuhlinzwa. Ngeke isetshenziselwe izifo zesibindi nezinso, izilonda zesisu, uhlobo lokuqunjelwa kwe-gastritis.
Ukuphendula okuvame kakhulu kufaka phakathi:
- i-leukopenia, thrombocytopenia;
- Ubuhlungu be-angina, ukwehlisa umfutho wegazi, izinhlungu zenhliziyo, ukubukeka kwe-arrhythmias;
- ubomvu besikhumba sobuso, i-angioedema, ukulunywa, ukushaqeka kwe-anaphylactic, i-urticaria;
- ukwehla kwesifiso sokudla, isifo sohudo, isicanucanu, ukuhlanza, usizi esiswini;
- ukuvela kwe-cholestatic hepatitis, ukwanda kwe-cholecystitis;
- ikhanda, imisipha, ukuphazamiseka kokulala, ukukhathazeka, isiyezi;
- ukungaboni kahle
- ukopha kwe-etiologies ehlukahlukene.
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Indlela yokudedelwa kwePentoxifylline ngamathebulethi, ama-ampoules anesixazululo somjovo. Qala ukuthatha umuthi ngomthamo wama-200 mg. Inkambo yokwelapha yinyanga. I-Pentoxifylline kuma-ampoules ibekelwa izifo ezinzima zezitho zangaphakathi noma inkambo yalesi sifo ngesimo esibi. Bafaka umuthi emthanjeni noma emsipha.
Ngokusebenzisana kwezidakamizwa zePentoxifylline ngama-anticoagulants kanye nemithi ye-antihypertensive, umphumela wokugcina uyathuthukiswa.
Ukusetshenziswa kwalo muthi ezigulini ezinesifo sikashukela kungaholela ekwenyukeni kokwehlisa ushukela kwezidakamizwa ze-antidiabetic futhi kungaze kubangele ukuthuthukiswa kokuphendula kwe-hypoglycemic.
I-Pentoxifylline analogues ifaka:
- I-Radomin.
- Trental.
- Dibazole
- I-Agapurin.
- Izimbali.
Umenzi walo muthi yi-Ozon Farm LLC, eRussia.
Isici seTrental
I-Trental ngumenzeli we-vasodilating, isakhi esiyinhloko saso yi-pentoxifylline. Ngaphezu kwalokho, ukwakheka kufaka phakathi izakhi ezingeziwe: isitashi, i-lactose, i-talc, i-silicon dioxide, i-sodium hydroxide, i-titanium dioxide, i-magnesium stearate.
Umuthi unomphumela we-vasodilating, normalizing ukuhamba kwegazi, uthuthukisa ukuphefumula kwamaselula. Isetshenziselwa i-frostbite, ukuphazamiseka kwengqondo, ukuphazamiseka kokujikeleza ku-choroid yeso nobuchopho.
I-Trental isiza umzimba ukuba ululame ngokushesha ngemuva kokushaywa unhlangothi, ithuthukise isimo nge-post-thrombotic kanye ne-ischemic syndrome, futhi inciphise izinhlungu nokuncipha emisipha yethole.
Umuthi ukhonjiswa ekwelapheni lezi zifo ezilandelayo:
- i-atherosclerotic encephalopathy;
- ischemic cerebral stroke;
- i-encirchalatory encephalopathy;
- ukwephulwa kokujikeleza kwegazi ngokumelene nesizinda sikashukela i-mellitus, isifo sokuqina kwemithambo yegazi, ukuwohloka kwe-endarteritis;
- ukuphazamiseka kwezicubu ze-trophic;
- i-arthrosis;
- ukwehluleka okujikelezayo kokujikeleza kwe-retina;
- i-vascular pathology yendlebe yangaphakathi;
- isifuba somoya;
- imithambo ye-varicose;
- gangren
- ukukhulisa potency.
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I-Trental yezidakamizwa inomphumela we-vasodilating, ibale ukuhamba kwegazi, ithuthukisa ukuphefumula kwamaselula.
Umuthi lo unezimpawu eziningi eziphikisayo. Kuyenqatshelwa ukuthatha kumacala alandelayo:
- ukungabekezelelani komuntu ngamunye ezingxenyeni zomuthi;
- infarction yakamuva myocardial;
- i-porphyria;
- ukopha kwangaphandle noma kwangaphakathi;
- ukushaya kwe-hemorrhagic;
- ukuphefumula kwe-capillary emehlweni;
- ukukhulelwa nokuqunjelwa;
- ukuphazamiseka kwesigqi senhliziyo;
- i-coronary or cerebral arteriossteosis;
- umfutho wegazi ophansi.
Kuvunyelwe ukuyisebenzisa ngasikhathi sinye ngamavithamini nemifino yokudla yemifino.
Ukuthatha i-Trental kungadala ukukhula kwemiphumela emibi engafuneki. Kungaba:
- iminyakazo
- Ukukhathazeka
- isiyezi, ikhanda, ukuphazamiseka kokulala;
- i-hyperemia yesikhumba;
- i-pancytopenia;
- ukwehlisa umfutho wegazi;
- ukungaboni kahle
- umlomo owomile
- ukuqhubeka kwe-angina;
- i-arrhythmia, i-Cardialgia, i-angina pectoris, i-tachycardia;
- i-thrombocytopenia;
- ukwehla kwesifiso sokudla;
- i-atony yamathumbu.
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I-Trental itholakala kumathebulethi nezixazululo ezifakelwayo. Umthamo omkhulu wansuku zonke yi-1.2 g. Uma uxhumana nezidakamizwa ezithile, ungavusa umphumela wazo. Lokhu kufaka phakathi ama-nitrate, ama-inhibitors, ama-thrombolytics, ama-anticoagulants, nama-antibiotics. Mhlawumbe inhlanganisela yokuvuselela izicubu zomzimba.
Analogs of Trental:
- I-Pentoxifylline.
- IPentamon.
- Izimbali.
Umenzi walo muthi yiSanofi India Limited, eNdiya.
Ukuqhathanisa kwePentoxifylline neTrental
Le mishanguzo i-analogues. Kunokufana okuningi, kepha kunomehluko.
Imiphi imikhiqizo efanayo
Ingxenye eyinhloko yeTrental nePentoxifylline iyafana - pentoxifylline. Zombili lezi zidakamizwa zikhombisa ukusebenza okufanayo ekwelapheni ukusakazeka kokujikeleza kwe-peripheral futhi zisetshenziselwa ukuqeda i-lameness.
Imithi inomphumela ofanayo ekwelashweni kwe-vascular pathologies. Zibekiwe njengezindlela eziphambili zokusiza ukususa imiphumela yokuhlaselwa yisifo sohlangothi kubantu. Kunconywa njengezidakamizwa zokuvimbela uma kunobungozi obukhulu bokuqothuka kwe-myocardial. I-Trental nePentoxifylline zinenombolo enkulu ye-contraindication nemiphumela emibi.
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IPentoxifylline neTrental zichazwe njengezindlela eziphambili zokususa imiphumela yokuhlaselwa yisifo sohlangothi kubantu.
Uyini umehluko
Umehluko wezidakamizwa yi-bioavailability. Ku-Trental, kungama-90-93%, kuPentoxifylline - 89-90%. Ukuphila kwengxenye yomenzeli wokuqala amahora angama-1-2, owesibili - amahora angama-2,5. Banabakhiqizi abahlukile.
Yikuphi okushibhile
IPentoxifylline ishibhile kakhulu. Izindleko zayo zingama-ruble angama-25-100. Intengo ye-Trental - ama-ruble ayi-160-1250.
Yikuphi okungcono - Pentoxifylline noma Trental
Ukukhetha ukuthi yisiphi isidakamizwa okufanele sikunikeze - I-Pentoxifylline noma i-Trental, udokotela uhlola isimo sesiguli, unaka isigaba sesifo, izinkomba kanye ne-contraindication. Ngokuphikisana nesizinda sokwelashwa ngeTrental, ukujikeleza kwegazi kubuyiselwa ngokushesha okukhulu. Ngokuphathwa kwe-intravenous, lesi sidakamizwa sivame ukubekwa njengokuthi sisebenze kakhudlwana futhi siphephile.
Ukubuyekezwa kweziguli
UMarina, oneminyaka engama-60, u-Inza: "Sekuyisikhathi eside ngihlushwa imithambo ye-varicose. Muva nje, kwaqhamuka isilonda esivele sivele emlenzeni wami esingakwazi ukwelapha utho. Udokotela wayala ukuthi abesehlise i-Trental. Ngemuva kwenqubo yesihlanu, isilonda sathuthuka futhi isilonda sambozwa ngogqwala ngasekupheleni kokwelashwa. Akukho kusabela okubi okwenzekile. "
UValentina, oneminyaka engama-55, uSaratov: "Udokotela usekutholele isikhathi eside ukuphazamiseka kwemithambo yegazi emithanjeni ye-popliteal and females. Muva nje, unikeze iPentoxifylline. Ngemuva kwenkambo yokwelashwa, isimo sakhe saba ngcono."
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Imithi Pentoxifylline neTrental inomphumela ofanayo ekwelashweni kwe-vascular pathologies.
Odokotela babuyekeza ngePentoxifylline, Trental
UDmitry, phlebologist: "Nsuku zonke ngamukela iziguli ezinokuphazanyiswa kwe-microcirculatory circul. Ngenxa yalokhu, ziba nezilonda ezikhuluphayo, isikhumba soma futhi sibe buthaka. Ukubuyisela i-microcirculation, nginquma iTrental noma iPentoxifylline yeziguli. yize kubiza kakhulu. "
U-Oleg, i-phlebologist: "IPentoxifylline inomphumela omuhle wokwelapha uma kunosongo lwe-thrombosis. Esikhundleni salokho, ngivame ukunquma iTrental, ekhombisa umphumela ofanayo. Le mithi ingahlanganiswa ne-venotonics yangaphandle."